SCHEMBL5879323

SCHEMBL5879323

O=C1C=C(c2c[nH]c3ccccc23)C(=O)O1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 1/20 0.58
PTPRF P10586 1/20 0.58
PTPN1 P18031 1/20 0.58
CDC25B P30305 1/20 0.58
SIRT2 Q8IXJ6 3/20 0.57
PRKCB P05771 3/20 0.57
PRKCA P17252 2/20 0.57
PRKD3 O94806 1/20 0.57
CCNB2 O95067 1/20 0.57
CCNE2 O96020 1/20 0.57
ABL1 P00519 1/20 0.57
PRKCG P05129 1/20 0.57
CDK1 P06493 1/20 0.57
PIM1 P11309 1/20 0.57
CDK4 P11802 1/20 0.57
CCNB1 P14635 1/20 0.57
PRKACA P17612 1/20 0.57
PRKACG P22612 1/20 0.57
PRKACB P22694 1/20 0.57
CCND1 P24385 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7951074 0.80 PTPN1 (0.73) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL8314810 0.80 TDO2 (0.49) CCNE2CDK4PRKACAPRKACGPRKACB
SCHEMBL7197287 0.77 PRKCB (0.68) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL29771997 0.75 PRKCB (0.65) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL1158441 0.75 PTPRC (0.60) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL2193383 0.75 PRKCB (0.65) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL1202543 0.74 IMPDH2 (0.63) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL8992461 0.73 PTPN1 (1.00) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL6824529 0.73 PTPRC (0.55) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL9572016 0.73 PTPN1 (0.77) PTPRCPTPRFPTPN1CDC25BSIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111978298-A Bis-indole maleimide fluorescence sensor containing aromatic amide group 广东石油化工学院 2020-11-24 CN claimed
CN-111978298-A Bis-indole maleimide fluorescence sensor containing aromatic amide group 广东石油化工学院 2020-11-24 CN disclosed
CN-101812097-A Indole carbazole and bisindole maleimide alkaloid and its production and application OCEAN UNIV CHINA 2010-08-25 CN disclosed
US-7151108-B2 Anticarcinogenic, antiproliferative, and antitumor agents LES LABORATORIES SERVIER (FR) 2006-12-19 US disclosed
EP-1411057-B1 [3,4-a:3,4-c]carbazole derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2005-04-27 EP disclosed
US-20040077672-A1 Anticarcinogenic, antiproliferative, and antitumor agents LES LABORATOIRES SERVIER (FR) 2004-04-22 US disclosed
EP-1411057-A1 [3,4-a:3,4-c]carbazole derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2004-04-21 EP disclosed
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP disclosed
US-5547976-A VIRICIDES, HERPES VIRUS, CYTOMEGALOVIRUS; CARDIOVASCULAR DISORDERS BURROUGHS WELLCOME CO. (US) 1996-08-20 US disclosed
EP-0630241-A1 INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1994-12-28 EP disclosed
WO-1993018765-A1 INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1993-09-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040077672-A1 Anticarcinogenic, antiproliferative, and antitumor agents XDH, TOP2A, TOP1 PTPRC 2403/4885PTPRF 1942/4885PTPN1 531/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.