SCHEMBL6498480

SCHEMBL6498480

CCCOC(C(=O)O)C(CNC(=O)c1nc(-c2ccccc2Cl)sc1C)c1ccc(OC)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSA P10619 2/20 0.39
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR2A P28223 5/20 0.35
HTR2C P28335 5/20 0.35
SLC6A4 P31645 5/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MGAM O43451 1/20 0.34
GAA P10253 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
TP53 P04637 3/20 0.34
LMNA P02545 3/20 0.33
MAPT P10636 2/20 0.33
P2RX7 Q99572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6505584 0.82 DGAT1 (0.38) ALDH1A1SMN1; SMN2NPC1RAB9AL3MBTL1
SCHEMBL6496508 0.82 FFAR2 (0.35) CTSAALDH1A1SMN1; SMN2HTR2CNPC1
SCHEMBL6496054 0.73 KDM4E (0.40) ALDH1A1SMN1; SMN2CYP2C19NPC1RAB9A
SCHEMBL6495786 0.73 NPC1 (0.38) ALDH1A1SMN1; SMN2NPC1RAB9AGAA
SCHEMBL7684255 0.73 SHMT1 (0.40) CTSAALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL6498475 0.73 PPARA (0.46) ALDH1A1LMNAMAPT
SCHEMBL6505070 0.72 TRPV1 (0.35) ALDH1A1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL6503799 0.71 EGLN2 (0.35) ALDH1A1SMN1; SMN2NPC1TP53MAPT
SCHEMBL6502680 0.70 CDC7 (0.41) SMN1; SMN2NPC1RAB9ATP53LMNA
SCHEMBL6503268 0.69 NPC1 (0.60) ALDH1A1SMN1; SMN2CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed