SCHEMBL6972122

SCHEMBL6972122

CC(C)c1nc(C(C)OCc2ccccc2)n(Cc2ccccc2[N+](=O)[O-])c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
ACHE P22303 1/20 0.32
DHODH Q02127 1/20 0.32
CASP1 P29466 1/20 0.32
CASP4 P49662 1/20 0.32
CASP5 P51878 1/20 0.32
MAPT P10636 1/20 0.32
NPC1 O15118 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
RAB9A P51151 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
CTSB P07858 1/20 0.31
CCR5 P51681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962626 0.84 AGTR1 (0.34) PIN1TDP1DHODHCASP1CASP4
SCHEMBL6964071 0.80 ALDH1A1 (0.35) TDP1ACHECASP1CASP4CASP5
SCHEMBL6972629 0.79 AGTR1 (0.37) TDP1DHODHCASP1CASP4CASP5
SCHEMBL6960943 0.77 AGTR1 (0.35) TDP1ALDH1A1KDM4ELMNACCR5
SCHEMBL6969339 0.72 ALDH1A1 (0.36) TDP1NPC1CYP1A2CYP2C9RAB9A
SCHEMBL7084809 0.71 TDP1 (0.33) TDP1
SCHEMBL14439828 0.71 TDP1 (0.40) TDP1DHODHMAPTNPC1RAB9A
SCHEMBL7078850 0.70 TDP1 (0.32) TDP1MAPTALDH1A1LMNA
SCHEMBL6969396 0.69 TDP1 (0.37) TDP1
SCHEMBL6966496 0.68 VCP (0.37) TDP1DHODHMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed