SCHEMBL6985295

SCHEMBL6985295

N#Cc1ccc(CCC(=O)N2CCCc3cccc(S(=O)(=O)NCc4ccccc4)c32)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.45
NSD2 O96028 1/20 0.43
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
KMT2A Q03164 2/20 0.41
HTT P42858 1/20 0.41
PRMT1 Q99873 1/20 0.39
CYP19A1 P11511 2/20 0.39
TP53 P04637 2/20 0.39
POLB P06746 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
OPRK1 P41145 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
FPR1 P21462 2/20 0.37
FPR2 P25090 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986981 0.89 MCL1 (0.40) MEN1ALDH1A1KMT2AFPR1FPR2
SCHEMBL6983751 0.85 NR3C1 (0.40) MAPTMEN1ALDH1A1KMT2AFPR1
SCHEMBL6980994 0.84 RXRA (0.43) MAPTMEN1ALDH1A1KMT2ATP53
SCHEMBL6985290 0.82 ALDH1A1 (0.58) MAPTMEN1ALDH1A1LMNAKMT2A
SCHEMBL6985566 0.81 PARP14 (0.40) MAPTMEN1ALDH1A1KMT2ATP53
SCHEMBL6985322 0.81 GAA (0.41) MAPTMEN1ALDH1A1LMNAKMT2A
SCHEMBL6987632 0.80 ALDH1A1 (0.39) MAPTMEN1ALDH1A1LMNAKMT2A
SCHEMBL6977890 0.80 SLC16A3 (0.46) MEN1ALDH1A1KMT2APOLB
SCHEMBL6986002 0.79 RXRA (0.45) MAPTMEN1ALDH1A1LMNAKMT2A
SCHEMBL6986817 0.79 THRB (0.42) MAPTALDH1A1LMNAKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed