SCHEMBL7225481

SCHEMBL7225481

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Oc2ccccc2)o1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.45
MAPT P10636 2/20 0.45
MAPK1 P28482 1/20 0.45
ALDH1A1 P00352 2/20 0.40
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
KLKB1 P03952 1/20 0.37
MMP2 P08253 1/20 0.37
MMP7 P09237 1/20 0.37
MMP9 P14780 1/20 0.37
MMP13 P45452 1/20 0.37
SLC6A4 P31645 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225739 0.90 ALDH1A1 (0.45) NPSR1MAPTMAPK1ALDH1A1SLC6A4
SCHEMBL7224670 0.90 LMNA (0.43) NPSR1MAPTMAPK1ALDH1A1SLC6A3
SCHEMBL7233832 0.87 SLC6A3 (0.42) NPSR1MAPTMAPK1ALDH1A1MMP13
SCHEMBL7226375 0.87 MAPT (0.48) NPSR1MAPTMAPK1ALDH1A1SLC6A4
SCHEMBL7232058 0.86 NPSR1 (0.40) NPSR1MAPTMAPK1ALDH1A1SLC6A4
SCHEMBL7230399 0.86 MAPT (0.36) NPSR1MAPTMAPK1ALDH1A1SLC6A4
SCHEMBL7225022 0.85 NPC1 (0.42) NPSR1MAPTMAPK1ALDH1A1HTR3E
SCHEMBL7125195 0.84 MMP2 (0.36) NPSR1ALDH1A1HTR3EHTR3BHTR3A
SCHEMBL7232127 0.83 SLC9A1 (0.48) MAPTMAPK1ALDH1A1HTR3EHTR3B
SCHEMBL7233162 0.83 HTR3E (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed