SCHEMBL7352017

SCHEMBL7352017

O=C(CCN1CCC2(CCCC2)CC1)c1ccc(I)cc1F

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.44
ACKR3 P25106 3/20 0.39
SIGMAR1 Q99720 1/20 0.37
HTR1A P08908 2/20 0.36
ADRA1B P35368 2/20 0.36
MAP2K2 P36507 2/20 0.36
MAP2K1 Q02750 2/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
ALDH1A1 P00352 4/20 0.35
KMT2A Q03164 3/20 0.35
MAPK1 P28482 1/20 0.35
GFER P55789 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352126 0.87 ALDH1A1 (0.47) DRD2ACKR3MAP2K2MAP2K1ALDH1A1
SCHEMBL7348115 0.86 DRD2 (0.47) DRD2ACKR3SIGMAR1HTR1AMAP2K2
SCHEMBL7353482 0.85 DRD2 (0.44) DRD2ACKR3SIGMAR1HTR1AADRA1B
SCHEMBL7350499 0.83 DRD2 (0.44) DRD2ACKR3SIGMAR1HTR1AADRA1B
SCHEMBL7351979 0.78 DRD2 (0.44) DRD2ACKR3SIGMAR1HTR1AADRA1B
SCHEMBL7352192 0.74 DRD2 (0.62) DRD2SIGMAR1HTR1AADRA1BKMT2A
SCHEMBL7354949 0.73 HTR1A (0.34) DRD2SIGMAR1HTR1AADRA1B
SCHEMBL7344816 0.73 MAPT (0.40) ACKR3MAP2K2MAP2K1ALDH1A1KMT2A
SCHEMBL7344636 0.72 DRD2 (0.47) DRD2ACKR3HTR1AALDH1A1KMT2A
SCHEMBL7348412 0.71 SMN1; SMN2 (0.48) ACKR3ALDH1A1KMT2AMAPK1GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0972764-A1 Aminoalcohols and aminoketones as CNS active agents Universita Degli Studi di Firenze (IT) 2000-01-19 EP claimed
EP-0972764-A1 Aminoalcohols and aminoketones as CNS active agents Universita Degli Studi di Firenze (IT) 2000-01-19 EP disclosed