SCHEMBL744735

SCHEMBL744735

COc1cc(C(=O)O)c(-c2ccc3cc4c(ccc5cc6cc7ccccc7cc6cc54)cc3c2)cc1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.48
HPGD P15428 4/20 0.48
ALDH1A1 P00352 4/20 0.48
ACMSD Q8TDX5 2/20 0.46
HSD17B10 Q99714 2/20 0.44
ERN1 O75460 1/20 0.44
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
MCL1 Q07820 1/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL742865 0.86 ACMSD (0.54) ACMSDHSD17B10SLC6A2SLC6A4SLC6A3
SCHEMBL745519 0.77 ACMSD (0.49) ACMSDHSD17B10CYP2D6CYP2C9MCL1
SCHEMBL2527550 0.75 ERN1 (0.52) KDM4EHPGDALDH1A1HSD17B10ERN1
SCHEMBL27542885 0.71 ACMSD (0.62) KDM4EHPGDALDH1A1ACMSDSLC6A2
SCHEMBL24895096 0.71 KDM4E (0.59) KDM4EHPGDALDH1A1HSD17B10LMNA
SCHEMBL23143203 0.71 KDM4E (0.66) KDM4EHPGDALDH1A1ACMSDHSD17B10
SCHEMBL9534725 0.71 KDM4E (0.66) KDM4EHPGDALDH1A1ACMSDHSD17B10
SCHEMBL10873515 0.70 ERN1 (0.58) KDM4EHPGDALDH1A1ACMSDHSD17B10
SCHEMBL743927 0.69 CA12 (0.49) KDM4EHPGDALDH1A1HSD17B10ERN1
SCHEMBL30746762 0.69 MAPT (0.47) KDM4EHPGDALDH1A1HSD17B10ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 74 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486404-A1 METABOLIC BIOMARKERS OF DRUG-INDUCED CARDIOTOXICITY Wisconsin Alumni Research Foundation (US) 2012-08-15 EP claimed
WO-2011044253-A1 METABOLIC BIOMARKERS OF DRUG-INDUCED CARDIOTOXICITY WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2011-04-14 WO claimed
US-20110081675-A1 Metabolic Biomarkers Of Drug-Induced Cardiotoxicity WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2011-04-07 US claimed
EP-4729063-A2 TREATMENT OF CANCER USING COENZYME Q10 COMBINATION THERAPIES BPGbio, Inc. (US) 2026-04-22 EP disclosed
US-20260091003-A1 METHODS OF TREATMENT OF TEMOZOLOMIDE-RESISTANT GLIOMA USING COENZYME Q10 BPGBIO INC (US) 2026-04-02 US disclosed
US-20260034073-A1 COMBINATION THERAPY OF COENZYME Q10 AND RADIATION FOR TREATMENT OF GLIOMA BPGBIO INC (US) 2026-02-05 US disclosed
EP-2983654-B1 TREATMENT OF CANCER USING COENZYME Q10 COMBINATION THERAPIES BPGBIO INC (US) 2025-11-12 EP disclosed
US-12303471-B2 Methods of treatment of temozolomide-resistant glioma using coenzyme Q10 BPGBIO, INC. (US) 2025-05-20 US disclosed
US-12209285-B2 Methods for treatment of oncological disorders using an epimetabolic shifter (coenzyme Q10) BPGBIO, INC. (US) 2025-01-28 US disclosed
US-11452699-B2 Method of treating or preventing tumors of the central nervous system BERG LLC (US) 2022-09-27 US disclosed
US-20220202741-A1 METHODS OF TREATMENT OF TEMOZOLOMIDE-RESISTANT GLIOMA USING COENZYME Q10 BERG, KARA ANN 2022-06-30 US disclosed
WO-2011031503-A2 METHODS FOR TREATMENT OF A SARCOMA USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) CYTOTECH LABS, LLC (US) 2011-03-17 WO disclosed
US-20110027247-A1 METHODS FOR TREATMENT OF ONCOLOGICAL DISORDERS USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) BERG LLC 2011-02-03 US disclosed
US-20110020312-A1 METHODS FOR TREATMENT OF METABOLIC DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS BERG LLC 2011-01-27 US disclosed
WO-2010132440-A2 METHODS FOR TREATMENT OF ONCOLOGICAL DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS CYTOTECH LABS, LLC (US) 2010-11-18 WO disclosed
WO-2010132479-A2 METHODS FOR THE DIAGNOSIS OF METABOLIC DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS CYTOTECH LABS, LLC (US) 2010-11-18 WO disclosed
WO-2010132502-A2 METHODS FOR TREATMENT OF METABOLIC DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS CYTOTECH LABS, LLC (US) 2010-11-18 WO disclosed
WO-2010132507-A2 METHODS FOR TREATMENT OF DISEASE USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) CYTOTECH LABS, LLC (US) 2010-11-18 WO disclosed
EP-2230312-A1 Probe compound for detecting and isolating enzymes and means and methods using the same Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2010-09-22 EP disclosed
WO-2009052186-A1 METABOLOMICS-BASED IDENTIFICATION OF DISEASE-CAUSING AGENTS GEORGIA TECH RESEARCH CORPORATION (US) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12209285-B2 Methods for treatment of oncological disorders using an epimetabolic shifter (coenzyme Q10) SLC25A20, NDUFB10, NDUFA10 KDM4E 2057/4885HPGD 236/4885ALDH1A1 778/4885
US-20260034073-A1 COMBINATION THERAPY OF COENZYME Q10 AND RADIATION FOR TREATMENT OF GLIOMA VEGFA, NDUFA10, NDUFB10 KDM4E 1631/4885HPGD 334/4885ALDH1A1 455/4885
US-20220202741-A1 METHODS OF TREATMENT OF TEMOZOLOMIDE-RESISTANT GLIOMA USING COENZYME Q10 NDUFB10, NDUFA10, NDUFB5 KDM4E 554/4885HPGD 305/4885ALDH1A1 766/4885
US-20260091003-A1 METHODS OF TREATMENT OF TEMOZOLOMIDE-RESISTANT GLIOMA USING COENZYME Q10 NDUFA10, NDUFB10, NDUFA5 KDM4E 828/4885HPGD 588/4885ALDH1A1 586/4885
US-20110020312-A1 METHODS FOR TREATMENT OF METABOLIC DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS PC, GLS2, PCK2 KDM4E 2944/4885HPGD 636/4885ALDH1A1 867/4885
US-20110027247-A1 METHODS FOR TREATMENT OF ONCOLOGICAL DISORDERS USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) SLC25A20, NDUFB10, NDUFA10 KDM4E 2057/4885HPGD 236/4885ALDH1A1 778/4885
US-11452699-B2 Method of treating or preventing tumors of the central nervous system NDUFB10, NDUFA10, COQ8A KDM4E 3221/4885HPGD 337/4885ALDH1A1 1181/4885
US-12303471-B2 Methods of treatment of temozolomide-resistant glioma using coenzyme Q10 NDUFB10, NDUFA10, NDUFB5 KDM4E 554/4885HPGD 305/4885ALDH1A1 766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.