SCHEMBL742865

SCHEMBL742865

O=C(O)c1cc(O)c(O)cc1-c1ccc2cc3c(ccc4cc5cc6ccccc6cc5cc43)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACMSD Q8TDX5 5/20 0.54
MCL1 Q07820 3/20 0.49
XDH P47989 1/20 0.45
SLC22A12 Q96S37 1/20 0.45
LCK P06239 1/20 0.44
ALOX5 P09917 1/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
SOS1 Q07889 2/20 0.42
HIF1A Q16665 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
GRIN2D O15399 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
TP53 P04637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HDAC4 P56524 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL744735 0.86 KDM4E (0.48) ACMSDMCL1ALOX5CYP2D6CYP2C9
SCHEMBL745519 0.84 ACMSD (0.49) ACMSDMCL1XDHSLC22A12CYP1A2
SCHEMBL27542885 0.78 ACMSD (0.62) ACMSDMCL1CYP1A2CYP2C19SOS1
SCHEMBL1247836 0.74 ACMSD (0.63) ACMSDMCL1XDHSLC22A12LCK
SCHEMBL12892157 0.73 MCL1 (0.74) ACMSDMCL1XDHSLC22A12GRIN2D
SCHEMBL19688783 0.72 NR4A1 (0.56) ACMSDMCL1SOS1HSD17B10LDHA
SCHEMBL3368675 0.72 ALDH1A1 (0.62) ACMSDCYP1A2CYP2C19SOS1HIF1A
SCHEMBL29618929 0.72 SLC6A2 (0.66) ACMSDMCL1CYP1A2CYP2C19SOS1
SCHEMBL84188 0.72 SLC6A2 (0.66) ACMSDMCL1CYP1A2CYP2C19SOS1
SCHEMBL30610922 0.72 SLC6A2 (0.66) ACMSDMCL1CYP1A2CYP2C19SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4729063-A2 TREATMENT OF CANCER USING COENZYME Q10 COMBINATION THERAPIES BPGbio, Inc. (US) 2026-04-22 EP disclosed
US-20260091003-A1 METHODS OF TREATMENT OF TEMOZOLOMIDE-RESISTANT GLIOMA USING COENZYME Q10 BPGBIO INC (US) 2026-04-02 US disclosed
US-20260034073-A1 COMBINATION THERAPY OF COENZYME Q10 AND RADIATION FOR TREATMENT OF GLIOMA BPGBIO INC (US) 2026-02-05 US disclosed
EP-2983654-B1 TREATMENT OF CANCER USING COENZYME Q10 COMBINATION THERAPIES BPGBIO INC (US) 2025-11-12 EP disclosed
US-12303471-B2 Methods of treatment of temozolomide-resistant glioma using coenzyme Q10 BPGBIO, INC. (US) 2025-05-20 US disclosed
US-12209285-B2 Methods for treatment of oncological disorders using an epimetabolic shifter (coenzyme Q10) BPGBIO, INC. (US) 2025-01-28 US disclosed
US-11452699-B2 Method of treating or preventing tumors of the central nervous system BERG LLC (US) 2022-09-27 US disclosed
US-20220202741-A1 METHODS OF TREATMENT OF TEMOZOLOMIDE-RESISTANT GLIOMA USING COENZYME Q10 BERG, KARA ANN 2022-06-30 US disclosed
US-20220096399-A1 METHODS OF TREATMENT OF SOLID TUMORS USING COENZYME Q10 BERG LLC (US) 2022-03-31 US disclosed
US-20220096400-A1 METHODS FOR THE TREATMENT OF CANCER USING COENZYME Q10 IN COMBINATION WITH IMMUNE CHECKPOINT MODULATORS THLIVERIS, ANDREW T. 2022-03-31 US disclosed
US-20110064747-A1 METHODS FOR TREATMENT OF A SARCOMA USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) BERG PHARMA LLC 2011-03-17 US disclosed
WO-2011031503-A2 METHODS FOR TREATMENT OF A SARCOMA USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) CYTOTECH LABS, LLC (US) 2011-03-17 WO disclosed
US-20110027247-A1 METHODS FOR TREATMENT OF ONCOLOGICAL DISORDERS USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) BERG LLC 2011-02-03 US disclosed
US-20110020312-A1 METHODS FOR TREATMENT OF METABOLIC DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS BERG LLC 2011-01-27 US disclosed
WO-2010132440-A2 METHODS FOR TREATMENT OF ONCOLOGICAL DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS CYTOTECH LABS, LLC (US) 2010-11-18 WO disclosed
WO-2010132479-A2 METHODS FOR THE DIAGNOSIS OF METABOLIC DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS CYTOTECH LABS, LLC (US) 2010-11-18 WO disclosed
WO-2010132502-A2 METHODS FOR TREATMENT OF METABOLIC DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS CYTOTECH LABS, LLC (US) 2010-11-18 WO disclosed
WO-2010132507-A2 METHODS FOR TREATMENT OF DISEASE USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) CYTOTECH LABS, LLC (US) 2010-11-18 WO disclosed
EP-2230312-A1 Probe compound for detecting and isolating enzymes and means and methods using the same Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2010-09-22 EP disclosed
WO-2009052186-A1 METABOLOMICS-BASED IDENTIFICATION OF DISEASE-CAUSING AGENTS GEORGIA TECH RESEARCH CORPORATION (US) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12209285-B2 Methods for treatment of oncological disorders using an epimetabolic shifter (coenzyme Q10) SLC25A20, NDUFB10, NDUFA10 ACMSD 4565/4885MCL1 727/4885XDH 702/4885
US-20260034073-A1 COMBINATION THERAPY OF COENZYME Q10 AND RADIATION FOR TREATMENT OF GLIOMA VEGFA, NDUFA10, NDUFB10 ACMSD 4497/4885MCL1 1270/4885XDH 1868/4885
US-20220202741-A1 METHODS OF TREATMENT OF TEMOZOLOMIDE-RESISTANT GLIOMA USING COENZYME Q10 NDUFB10, NDUFA10, NDUFB5 ACMSD 4450/4885MCL1 1458/4885XDH 1020/4885
US-20220096400-A1 METHODS FOR THE TREATMENT OF CANCER USING COENZYME Q10 IN COMBINATION WITH IMMUNE CHECKPOINT MODULATORS NDUFA10, NDUFB10, NDUFA5 ACMSD 3675/4885MCL1 635/4885XDH 1414/4885
US-20260091003-A1 METHODS OF TREATMENT OF TEMOZOLOMIDE-RESISTANT GLIOMA USING COENZYME Q10 NDUFA10, NDUFB10, NDUFA5 ACMSD 3722/4885MCL1 1587/4885XDH 1397/4885
US-20110020312-A1 METHODS FOR TREATMENT OF METABOLIC DISORDERS USING EPIMETABOLIC SHIFTERS, MULTIDIMENSIONAL INTRACELLULAR MOLECULES, OR ENVIRONMENTAL INFLUENCERS PC, GLS2, PCK2 ACMSD 3506/4885MCL1 2687/4885XDH 1442/4885
US-20110027247-A1 METHODS FOR TREATMENT OF ONCOLOGICAL DISORDERS USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) SLC25A20, NDUFB10, NDUFA10 ACMSD 4565/4885MCL1 727/4885XDH 702/4885
US-11452699-B2 Method of treating or preventing tumors of the central nervous system NDUFB10, NDUFA10, COQ8A ACMSD 3220/4885MCL1 2402/4885XDH 898/4885
US-12303471-B2 Methods of treatment of temozolomide-resistant glioma using coenzyme Q10 NDUFB10, NDUFA10, NDUFB5 ACMSD 4450/4885MCL1 1458/4885XDH 1020/4885
US-20220096399-A1 METHODS OF TREATMENT OF SOLID TUMORS USING COENZYME Q10 NDUFB10, NDUFA10, NDUFB5 ACMSD 4608/4885MCL1 577/4885XDH 984/4885
US-20110064747-A1 METHODS FOR TREATMENT OF A SARCOMA USING AN EPIMETABOLIC SHIFTER (COENZYME Q10) NDUFB10, SDHB, SDHA ACMSD 3939/4885MCL1 1248/4885XDH 1762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.