SCHEMBL7475491

SCHEMBL7475491

CCc1ccc(C(=O)NC2(c3ccccc3)C(=O)NC(=O)NC2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.45
HDAC6 Q9UBN7 2/20 0.43
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
KLF5 Q13887 1/20 0.41
MMP9 P14780 3/20 0.40
MMP8 P22894 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
SLC16A3 O15427 1/20 0.40
PPARA Q07869 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
MMP2 P08253 2/20 0.40
POLB P06746 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482004 0.86 ALDH1A1 (0.46) HDAC6ALDH1A1GAAMMP9MMP8
SCHEMBL7478795 0.85 LMNA (0.45) HDAC6ALDH1A1NPC1RAB9AGAA
SCHEMBL7481304 0.84 NPC1 (0.49) PLK1ALDH1A1NPC1RAB9AGAA
SCHEMBL7480698 0.83 AKR1B1 (0.48) ALDH1A1NPC1RAB9AGAAMMP9
SCHEMBL7475641 0.82 PTGS2 (0.44) HDAC6ALDH1A1NPC1RAB9AGAA
SCHEMBL7474643 0.82 ALDH1A1 (0.45) ALDH1A1NPC1RAB9AMMP9TDP1
SCHEMBL7477845 0.82 MMP9 (0.42) ALDH1A1MMP9MMP8TDP1MMP2
SCHEMBL7482164 0.82 MMP2 (0.49) PLK1ALDH1A1NPC1RAB9AGAA
SCHEMBL7484780 0.82 MMP9 (0.46) PLK1NPC1RAB9AMMP9MMP8
SCHEMBL7470955 0.80 HTT (0.46) ALDH1A1RAB9AGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472396-B1 Barbituric acid derivatives, processes for their production and pharmaceutical agents containing these compounds ROCHE DIAGNOSTICS GMBH (DE) 2002-10-29 US claimed
EP-0869947-B1 BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 2002-10-23 EP disclosed