SCHEMBL7546196

SCHEMBL7546196

Cc1ccsc1CC(=O)c1ccnc(N)c1C(=O)Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
KDM6B O15054 1/20 0.38
KDM4A O75164 1/20 0.38
KDM5C P41229 1/20 0.38
KDM4D Q6B0I6 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
SLCO1B1 Q9Y6L6 1/20 0.38
ALOX5 P09917 1/20 0.37
GSK3B P49841 1/20 0.35
PNP P00491 2/20 0.33
HSD11B1 P28845 1/20 0.32
RIPK1 Q13546 1/20 0.32
NPC1 O15118 1/20 0.31
PPARG P37231 1/20 0.31
RAB9A P51151 1/20 0.31
NCOR2 Q9Y618 1/20 0.31
POLB P06746 1/20 0.31
NOS3 P29474 3/20 0.31
NOS2 P35228 3/20 0.31
LIMK1 P53667 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799100 0.89 KDM4E (0.44) KDM4EKDM6BKDM4AKDM5CKDM4D
SCHEMBL7600813 0.83
SCHEMBL7549098 0.79 RAB9A (0.41) GSK3BNPC1PPARGRAB9ANCOR2
SCHEMBL7546276 0.78 MEN1 (0.45) KDM4ENPC1NOS3NOS2
SCHEMBL7546252 0.77 TDP1 (0.32) PPARGNOS3NOS2TP53
SCHEMBL7545898 0.74 NAMPT (0.36) NPC1RAB9ANOS3NOS2LIMK1
SCHEMBL7548395 0.74 ALOX5 (0.38) ALOX5NPC1RAB9A
SCHEMBL9059987 0.74 SGMS2 (0.35) KDM4EKDM4CTP53
SCHEMBL9059311 0.72 NAPRT (0.34) KDM4EKDM6BKDM4AKDM5CKDM4D
SCHEMBL8799386 0.71 SHBG (0.44) KDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997049708-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1998-05-22 WO disclosed