SCHEMBL7656052

SCHEMBL7656052

COc1ccccc1-n1nc(-c2ccccc2)n(C)c1=O

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.54
ADORA3 P0DMS8 2/20 0.54
ADORA2A P29274 1/20 0.52
AVPR2 P30518 1/20 0.48
AVPR1A P37288 1/20 0.48
MGLL Q99685 1/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 1/20 0.46
APOBEC3G Q9HC16 1/20 0.46
TP53 P04637 1/20 0.45
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TSHR P16473 1/20 0.41
KCNN4 O15554 1/20 0.41
UGCG Q16739 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7659194 0.82 ALDH1A1 (0.51) ADORA2AMGLLALDH1A1KDM4EMAPT
SCHEMBL7656700 0.80 ADORA3 (0.47) ADORA1ADORA3ADORA2AAVPR2AVPR1A
SCHEMBL7660359 0.79 MGLL (0.44) ADORA2AMGLLALDH1A1MAPTTSHR
SCHEMBL7652883 0.79 OPRM1 (0.41) ADORA2AMGLLALDH1A1NPC1RAB9A
SCHEMBL7652394 0.79 HSD11B1 (0.45) ADORA2AMGLL
SCHEMBL7658070 0.79 NPC1 (0.44) MGLLALDH1A1NPC1RAB9ANPSR1
Dimethylamine SCHEMBL7656702 0.79 ADORA3 (0.48) ADORA1ADORA3ADORA2AAVPR2AVPR1A
SCHEMBL1784121 0.77 MGLL (0.46) ADORA1ADORA3ADORA2AMGLLALDH1A1
SCHEMBL7652545 0.77 ADORA3 (0.49) ADORA1ADORA3ADORA2AALDH1A1NPC1
Dimethylamine SCHEMBL7656223 0.76 MGLL (0.41) ADORA2AMGLLALDH1A1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492407-B2 NEUROPROTECTIVE ACTIVITY BOEHRINGER IMGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed