SCHEMBL7656700

SCHEMBL7656700

COc1ccccc1-n1nc(-c2ccccc2)n(CCN(C)C)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.47
ADORA1 P30542 2/20 0.47
ADORA2A P29274 1/20 0.45
TDP1 Q9NUW8 2/20 0.41
AVPR2 P30518 1/20 0.41
AVPR1A P37288 1/20 0.41
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
APOBEC3G Q9HC16 1/20 0.39
TSHR P16473 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
FABP3 P05413 1/20 0.38
MDM4 O15151 1/20 0.38
MDM2 Q00987 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRA1D P25100 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652938 0.85 ALDH1A1 (0.43) ADORA3ADORA2AALDH1A1KDM4ETSHR
SCHEMBL7656105 0.84 DRD2 (0.39) ADORA3ADORA2AALDH1A1KDM4ETSHR
SCHEMBL7652262 0.83 NOX4 (0.45) ADORA3ADORA2AALDH1A1KDM4ETSHR
SCHEMBL7653997 0.83 OPRM1 (0.38) ADORA3ADORA2AALDH1A1KDM4ETSHR
SCHEMBL7653733 0.83 NPC1 (0.40) ADORA3ALDH1A1KDM4ETSHRHPGD
SCHEMBL7656086 0.81 CTSK (0.45) ADORA3ADORA1ADORA2AALDH1A1KDM4E
Dimethylamine SCHEMBL7656702 0.81 ADORA3 (0.48) ADORA3ADORA1ADORA2AAVPR2AVPR1A
SCHEMBL7656052 0.80 ADORA1 (0.54) ADORA3ADORA1ADORA2AAVPR2AVPR1A
SCHEMBL7652889 0.80 CTSK (0.45) ADORA3ADORA1ADORA2AALDH1A1KDM4E
SCHEMBL7651062 0.79 CA1 (0.37) ADORA3ALDH1A1KDM4ETSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492407-B2 NEUROPROTECTIVE ACTIVITY BOEHRINGER IMGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed