SCHEMBL7709540

SCHEMBL7709540

CC(=O)N1CC(=S)C[C@H]1C(=O)O.NC(Cc1cccc(NC(=O)Cc2c(Cl)cccc2Cl)c1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
ACKR3 P25106 8/20 0.43
SLC7A5 Q01650 3/20 0.38
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
RECQL P46063 1/20 0.36
AGTR2 P50052 1/20 0.36
LMNA P02545 2/20 0.35
MAPT P10636 1/20 0.35
SIGMAR1 Q99720 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7905211 0.92 ITGB1 (0.43) ACKR3ITGB1ITGA4RECQLAGTR2
SCHEMBL7706489 0.85 NLRP3 (0.46) NOS3NOS1NOS2ACKR3SLC7A5
SCHEMBL7709242 0.84 NOS3 (0.47) NOS3NOS1NOS2SLC7A5
SCHEMBL7709457 0.83 NOS3 (0.43) NOS3NOS1NOS2ACKR3SLC7A5
SCHEMBL7703583 0.82 AGTR2 (0.40) SLC7A5ITGB1ITGA4AGTR2
SCHEMBL7905098 0.80 ITGB1 (0.50) ITGB1ITGA4
SCHEMBL6933788 0.79 AGTR2 (0.39) ITGB1ITGA4AGTR2
Phenylalanine SCHEMBL7906184 0.79 SLC7A5 (0.52) NOS3NOS1NOS2SLC7A5HDAC8
SCHEMBL6933976 0.78 ITGA4 (0.46) ITGB1ITGA4
SCHEMBL7896702 0.77 TPH1 (0.37) SLC7A5ITGB1ITGA4AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362204-B1 CONTROLLING IMMUNOLOGY; ANTIINFLAMMATORY AGENTS CELLTECH THERAPEUTICS, LTD (GB) 2002-03-26 US claimed
US-6362204-B1 CONTROLLING IMMUNOLOGY; ANTIINFLAMMATORY AGENTS CELLTECH THERAPEUTICS, LTD (GB) 2002-03-26 US disclosed