SCHEMBL7709242

SCHEMBL7709242

CC(=O)N1CC(=S)C[C@H]1C(=O)O.CC(C)(C)C(=O)Nc1cccc(CC(N)C(=O)O)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.47
NOS1 P29475 3/20 0.47
NOS2 P35228 3/20 0.47
SLC7A5 Q01650 5/20 0.41
NPY2R P49146 2/20 0.37
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
GRIA2 P42262 1/20 0.35
ALPI P09923 1/20 0.34
PKM P14618 1/20 0.34
PTGS1 P23219 1/20 0.34
XIAP P98170 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7906163 0.89 L3MBTL1 (0.36) SLC7A5NPY2RALPIPKMPTGS1
SCHEMBL7709540 0.84 NOS3 (0.43) NOS3NOS1NOS2SLC7A5
SCHEMBL7709457 0.83 NOS3 (0.43) NOS3NOS1NOS2SLC7A5
SCHEMBL7706489 0.82 NLRP3 (0.46) NOS3NOS1NOS2SLC7A5
Phenylalanine SCHEMBL7906184 0.82 SLC7A5 (0.52) NOS3NOS1NOS2SLC7A5ALPI
SCHEMBL7904116 0.77 SLC7A5 (0.45) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL7896693 0.77 ITGB1 (0.47)
SCHEMBL7905098 0.76 ITGB1 (0.50)
SCHEMBL6932583 0.76 PTPN1 (0.46) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL7908862 0.76 ALDH1A1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362204-B1 CONTROLLING IMMUNOLOGY; ANTIINFLAMMATORY AGENTS CELLTECH THERAPEUTICS, LTD (GB) 2002-03-26 US disclosed