SCHEMBL7938686

SCHEMBL7938686

O=C(C(=O)N(Cc1ccccn1)CC1CCCCC1)c1c[nH]c2cc(F)ccc12

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.38
KDR P35968 1/20 0.38
HAT1 O14929 1/20 0.37
EP300 Q09472 1/20 0.37
HPGD P15428 2/20 0.37
RECQL P46063 1/20 0.37
PKM P14618 3/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK14 Q16539 1/20 0.35
SLC6A9 P48067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3265771 0.87 MAPT (0.50) ALDH1A1TSHRKDRHPGDRECQL
SCHEMBL7982425 0.85 PKM (0.43) ALDH1A1HAT1EP300PKMROCK2
SCHEMBL7946315 0.83 MAPK14 (0.36) ALDH1A1PKMROCK2ROCK1KMT2A
SCHEMBL3263677 0.83 GABRA1 (0.45) ALDH1A1LMNAHAT1EP300HPGD
SCHEMBL3120950 0.81 ALDH1A1 (0.40) ALDH1A1TSHRPKMNPC1RAB9A
SCHEMBL4306639 0.81 MAPK14 (0.37) ALDH1A1PKMROCK2ROCK1KMT2A
SCHEMBL4304078 0.79 MAPK14 (0.43) ALDH1A1PKMROCK2ROCK1KMT2A
SCHEMBL4313368 0.78 ALDH1A1 (0.43) ALDH1A1HPGDRAB9AMAPK14
SCHEMBL4312756 0.78 HDAC1 (0.47) ALDH1A1LMNAPKMNPC1RAB9A
SCHEMBL4310271 0.77 ALDH1A1 (0.41) ALDH1A1ROCK2ROCK1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010035032-A1 CALCIUM ION CHANNEL MODULATORS & USES THEREOF LECTUS THERAPEUTICS LIMITED (GB) 2010-04-01 WO disclosed
WO-2009133387-A1 INDOLE- 3 -GLYOXYLAMIDE DERIVATIVES FOR USE AS CALCIUM ION CHANNEL MODULATORS LECTUS THERAPEUTICS LIMITED (GB) 2009-11-05 WO disclosed