SCHEMBL7962210

SCHEMBL7962210

COc1cccc(OC[C@H](O)CN2CCC(O)(c3cnc4ccccc4n3)CC2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.56
MAPT P10636 2/20 0.56
L3MBTL1 Q9Y468 2/20 0.55
KDM4E B2RXH2 2/20 0.54
GAA P10253 2/20 0.52
MAPK1 P28482 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
ACE2 Q9BYF1 1/20 0.49
KDR P35968 1/20 0.48
PRMT5 O14744 1/20 0.48
WDR77 Q9BQA1 1/20 0.48
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
RAD52 P43351 1/20 0.47
SCN1A P35498 1/20 0.47
SCN5A Q14524 1/20 0.47
SCN9A Q15858 1/20 0.47
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963018 0.87 TP53 (0.56) TP53MAPTL3MBTL1KDM4EGAA
SCHEMBL7962698 0.83 L3MBTL1 (0.46) L3MBTL1KDM4EGAAMAPK1SMN1; SMN2
SCHEMBL7962746 0.83 SMN1; SMN2 (0.47) MAPTL3MBTL1KDM4EMAPK1SMN1; SMN2
SCHEMBL7962212 0.82 ALDH1A1 (0.41) TP53MAPTKDM4ESMN1; SMN2MEN1
SCHEMBL7962207 0.82 ALDH1A1 (0.43) TP53MAPTL3MBTL1KDM4EMAPK1
SCHEMBL7953344 0.79 KDM4E (0.53) MAPTL3MBTL1KDM4EMAPK1SMN1; SMN2
SCHEMBL7965117 0.79 CYP1A2 (0.58) TP53MAPTGAASMN1; SMN2MEN1
Sulfuric Acid SCHEMBL7968960 0.78 ADORA2A (0.39) KDM4EGAASMN1; SMN2PRMT5WDR77
SCHEMBL7963395 0.77 LMNA (0.44) TP53MAPTKDM4ESMN1; SMN2MEN1
SCHEMBL7969553 0.76 L3MBTL1 (0.55) L3MBTL1KDM4ESMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed