SCHEMBL7965117

SCHEMBL7965117

O[C@@H](COc1ccc(Cl)cc1Cl)CN1CCC(O)(c2cnc3ccccc3n2)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.58
CYP2D6 P10635 1/20 0.58
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
USP2 O75604 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 2/20 0.47
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
F8 P00451 1/20 0.45
F5 P12259 1/20 0.45
TP53 P04637 1/20 0.45
ATM Q13315 1/20 0.43
ABCB1 P08183 6/20 0.43
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
IDE P14735 1/20 0.42
XBP1 P17861 1/20 0.42
PAX8 Q06710 1/20 0.42
HRH1 P35367 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7964392 0.87 CYP1A2 (0.58) CYP1A2CYP2D6MEN1KMT2AUSP2
SCHEMBL7965119 0.83 OPRM1 (0.39) CYP1A2CYP2D6MEN1KMT2ANPSR1
SCHEMBL7965112 0.81 LMNA (0.39) CYP1A2CYP2D6KMT2AUSP2NPSR1
SCHEMBL7963395 0.80 LMNA (0.44) CYP1A2CYP2D6MEN1KMT2ANPSR1
SCHEMBL7962698 0.79 L3MBTL1 (0.46) CYP2D6MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL7962210 0.79 TP53 (0.56) MEN1KMT2AMAPTSMN1; SMN2TP53
SCHEMBL7964941 0.78 CCR1 (0.45) CYP1A2MEN1KMT2ANPSR1MAPT
SCHEMBL7962746 0.77 SMN1; SMN2 (0.47) USP2HTTNPSR1MAPTSMN1; SMN2
Fumaric Acid SCHEMBL7966212 0.75 ABCB1 (0.51) MEN1KMT2AHTTMAPTSMN1; SMN2
SCHEMBL7965174 0.74 KMT2A (0.52) KMT2AMAPTSMN1; SMN2ABCB1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed