SCHEMBL7963392

SCHEMBL7963392

Cc1ccc(OCCC(O)N2CCC(O)(c3cnc4ccccc4n3)CC2)c2c1CCC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.35
ADRB1 P08588 3/20 0.35
CYP1A2 P05177 2/20 0.35
HIF1A Q16665 2/20 0.35
ADRA2A P08913 1/20 0.35
ADRB3 P13945 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
PMP22 Q01453 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXRA P19793 3/20 0.31
RXRB P28702 3/20 0.31
RXRG P48443 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7953681 0.86 ADRB2 (0.34) ADRB2ADRB1CYP1A2HIF1AADRA2A
SCHEMBL7963395 0.82 LMNA (0.44) ADRB2ADRB1CYP1A2HIF1AADRA2A
SCHEMBL7963401 0.81 ADRB2 (0.33) ADRB2ADRB1CYP1A2HIF1AADRA2A
SCHEMBL7965112 0.80 LMNA (0.39) CYP1A2KDM4ETP53CYP2D6TSHR
Fumaric Acid SCHEMBL7966209 0.79 MAPT (0.38) MEN1LMNAKMT2ANPSR1HCRTR1
Fumaric Acid SCHEMBL7966218 0.79 MAPT (0.38) MEN1LMNAKMT2ANPSR1HCRTR1
SCHEMBL7962207 0.78 ALDH1A1 (0.43) KDM4ETP53TSHRMEN1LMNA
SCHEMBL7962696 0.78 LTA4H (0.35) KDM4EMEN1LMNAKMT2AOPRM1
SCHEMBL7964944 0.77 MEN1 (0.30) MEN1KMT2A
Salicylic Acid SCHEMBL8133872 0.76 ABCB1 (0.32) KDM4ELMNAHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242450-B1 SUBSTITUTED PIPERIDINES ELI LILLY AND COMPANY 2001-06-05 US disclosed
WO-2000006166-A1 5-HT1F ANTAGONISTS ELI LILLY AND COMPANY (US) 2000-02-10 WO disclosed
EP-0976746-A1 5-HT1F antagonists ELI LILLY AND COMPANY (US) 2000-02-02 EP disclosed