SCHEMBL798232

SCHEMBL798232

O=Nc1ccc(O)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD17B1 P14061 4/20 0.38
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
HSD17B2 P37059 3/20 0.38
MGLL Q99685 3/20 0.38
SNCA P37840 1/20 0.38
CYP17A1 P05093 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP19A1 P11511 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 3/20 0.37
MAPT P10636 2/20 0.37
TSHR P16473 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4403906 0.78 CES2 (0.41) HSD17B10LMNACYP17A1CYP3A4CYP11B1
SCHEMBL3316934 0.78 PTGS2 (0.48) HSD17B10LMNAKDM4EALDH1A1HTT
SCHEMBL12228262 0.74 MAPT (0.40) HSD17B10LMNAKDM4ECYP3A4ALDH1A1
SCHEMBL1274361 0.74 ALDH1A1 (0.34) HSD17B10LMNACYP3A4ALDH1A1HTT
SCHEMBL29577999 0.74 ALDH1A1 (0.34) HSD17B10LMNACYP3A4ALDH1A1HTT
SCHEMBL4845445 0.74 TDP1 (0.49) KDM4EESR1ESR2ALDH1A1HTT
SCHEMBL25453075 0.73 KDM1A (0.37) HSD17B10LMNAKDM4ECYP3A4ALDH1A1
SCHEMBL639211 0.73 RAB9A (0.52) HSD17B10KDM4EHSD17B1ESR1ESR2
SCHEMBL11213671 0.73 PTGS1 (0.53) HSD17B10LMNAESR1ESR2CYP3A4
SCHEMBL18403872 0.73 ALOX15 (0.50) HSD17B10LMNAALDH1A1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100402487-C Method for preparing 2-fluoro-4-nitrophenol CHANGZHOU YETAI FINE CHEMICAL (CN) 2008-07-16 CN claimed
CN-1850778-A Method for preparing 2-fluoro-4-nitrophenol YETAI FINE CHEMICAL INST CHANG (CN) 2006-10-25 CN claimed
US-8329726-B2 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE INC. (CA) 2012-12-11 US disclosed
US-20120108628-A1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY Mirati Therapeutics, Inc. 2012-05-03 US disclosed
US-20120095234-A1 PROCESSES AND INTERMEDIATES FOR PREPARING FUSED HETEROCYCLIC KINASE INHIBITORS Mirati Therapeutics, Inc. 2012-04-19 US disclosed
US-20120083482-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE INC. 2012-04-05 US disclosed
US-8143305-B2 2,3-substituted indole derivatives for treating viral infections SCHERING CORPORATION (US) 2012-03-27 US disclosed
US-20120070413-A1 METHOD OF TREATING CANCER WITH SUBSTITUTED AMIDE DERIVATIVES KIM TAE-SEONG (US) 2012-03-22 US disclosed
US-8093264-B2 Fused heterocycles as inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE INC. (CA) 2012-01-10 US disclosed
US-20110104110-A1 SUBSTITUTED INDOLE DERIVATIVES AND METHODS OF USE THEREOF SHERING CORPORATION 2011-05-05 US disclosed
US-20110098293-A1 Inhibitors of Protein Tyrosine Kinase Activity OTSUKA PHARMACEUTICAL CO. LTD. (JP) 2011-04-28 US disclosed
US-20090286984-A1 Processes and intermediates for preparing fused heterocyclic kinase inhibitors Mirati Therapeutics, Inc. 2009-11-19 US disclosed
US-20090264440-A1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY Mirati Therapeutics, Inc. 2009-10-22 US disclosed
US-7547782-B2 Met kinase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2009-06-16 US disclosed
US-20080312232-A1 Substituted amide derivatives and methods of use AMGEN INC. (US) 2008-12-18 US disclosed
US-7442698-B2 Substituted heterocyclic compounds and methods of use AMGEN INC. (US) 2008-10-28 US disclosed
CN-100402487-C Method for preparing 2-fluoro-4-nitrophenol CHANGZHOU YETAI FINE CHEMICAL (CN) 2008-07-16 CN disclosed
CN-100402487-C Method for preparing 2-fluoro-4-nitrophenol CHANGZHOU YETAI FINE CHEMICAL (CN) 2008-07-16 CN disclosed
US-20080064718-A1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY METHYLGENE INC. (CA) 2008-03-13 US disclosed
CN-1850778-A Method for preparing 2-fluoro-4-nitrophenol YETAI FINE CHEMICAL INST CHANG (CN) 2006-10-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120095234-A1 PROCESSES AND INTERMEDIATES FOR PREPARING FUSED HETEROCYCLIC KINASE INHIBITORS MAP3K19, MAP3K9, MAP4K2 HSD17B10 2594/4885LMNA 3109/4885KDM4E 776/4885
US-20120083482-A1 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING HGF, MET, KDR HSD17B10 892/4885LMNA 4840/4885KDM4E 4651/4885
US-20090286984-A1 Processes and intermediates for preparing fused heterocyclic kinase inhibitors MAP3K19, MAP3K9, MAP4K2 HSD17B10 2594/4885LMNA 3109/4885KDM4E 776/4885
US-20090264440-A1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY HGF, ERBB2, MET HSD17B10 3782/4885LMNA 4752/4885KDM4E 2282/4885
US-20110104110-A1 SUBSTITUTED INDOLE DERIVATIVES AND METHODS OF USE THEREOF IDO1, IDO2, INMT HSD17B10 1083/4885LMNA 3284/4885KDM4E 1111/4885
US-20080312232-A1 Substituted amide derivatives and methods of use HGF, HGFAC, MET HSD17B10 922/4885LMNA 3752/4885KDM4E 3651/4885
US-20080064718-A1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY HGF, ERBB2, MET HSD17B10 3782/4885LMNA 4752/4885KDM4E 2282/4885
US-20120070413-A1 METHOD OF TREATING CANCER WITH SUBSTITUTED AMIDE DERIVATIVES HGF, HGFAC, MET HSD17B10 686/4885LMNA 3964/4885KDM4E 3048/4885
US-20120108628-A1 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY HGF, ERBB2, MET HSD17B10 3782/4885LMNA 4752/4885KDM4E 2282/4885
US-20110098293-A1 Inhibitors of Protein Tyrosine Kinase Activity ABL1, ERBB2, TYRO3 HSD17B10 4206/4885LMNA 4639/4885KDM4E 1254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.