SCHEMBL8043233

SCHEMBL8043233

NS(=O)(=O)c1ccc(-n2nnnc2Sc2nc(-c3ccccc3)cs2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.56
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA9 Q16790 3/20 0.47
CA12 O43570 1/20 0.47
CA5A P35218 1/20 0.47
CA5B Q9Y2D0 1/20 0.47
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
MMP2 P08253 1/20 0.42
CYP2C9 P11712 1/20 0.42
PTGS1 P23219 2/20 0.42
UBE2M P61081 1/20 0.41
DCUN1D1 Q96GG9 1/20 0.41
CA4 P22748 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050817 0.90 PTGS2 (0.57) PTGS2CA1CA2CA9CA12
SCHEMBL8044812 0.86 ALDH1A1 (0.52) MEN1MAPTHTTRAB9AKMT2A
SCHEMBL8034180 0.86 MAPT (0.49) PTGS2MEN1MAPTHTTKMT2A
SCHEMBL8043931 0.84 PTGS2 (0.43) PTGS2CA1CA2CA9CA12
SCHEMBL8046294 0.83 UBE2M (0.45) MAPTHTTRAB9AKMT2AUBE2M
SCHEMBL8045514 0.83 HPGD (0.54) MEN1MAPTHTTRAB9AKMT2A
SCHEMBL8032472 0.82 PTGS2 (0.48) PTGS2CA1CA2CA9CA12
SCHEMBL8042528 0.81 ALDH1A1 (0.45) MAPTHTTRAB9AKMT2AUBE2M
SCHEMBL8042159 0.81 RAB9A (0.47) PTGS2MEN1MAPTHTTRAB9A
SCHEMBL8044654 0.81 MAPT (0.44) PTGS2MEN1MAPTHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed