SCHEMBL8423

SCHEMBL8423

O=c1ccc2ccc(OCCCCN3CCN(c4cccc(Cl)c4Cl)CC3)cc2[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 18/20 1.00
HTR1A P08908 5/20 0.77
HTR2A P28223 5/20 0.77
DRD3 P35462 5/20 0.68
DRD4 P21917 4/20 0.68
ADRB2 P07550 2/20 0.68
ADRB1 P08588 2/20 0.68
ADRA2A P08913 2/20 0.68
ADRA2B P18089 2/20 0.68
ADRA2C P18825 2/20 0.68
DRD1 P21728 2/20 0.68
DRD5 P21918 2/20 0.68
SLC6A2 P23975 2/20 0.68
ADRA1D P25100 2/20 0.68
HTR1D P28221 2/20 0.68
HTR1B P28222 2/20 0.68
HTR2C P28335 2/20 0.68
SLC6A4 P31645 2/20 0.68
HTR7 P34969 2/20 0.68
ADRA1A P35348 2/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29549434 1.00 DRD2 (1.00) DRD2HTR1AHTR2ADRD3DRD4
SCHEMBL30552363 1.00 DRD2 (1.00) DRD2HTR1AHTR2ADRD3DRD4
Hydrochloric Acid SCHEMBL29365523 0.99 DRD2 (0.98) DRD2HTR1AHTR2ADRD3DRD4
Hydrochloric Acid SCHEMBL29923538 0.99 DRD2 (0.98) DRD2HTR1AHTR2ADRD3DRD4
SCHEMBL30964304 0.99 DRD2 (0.98) DRD2HTR1AHTR2ADRD3DRD4
SCHEMBL14587005 0.97 DRD2 (0.94) DRD2HTR1AHTR2ADRD3DRD4
SCHEMBL251904 0.96 DRD2 (1.00) DRD2HTR1AHTR2ADRD3DRD4
SCHEMBL253673 0.93 DRD2 (1.00) DRD2HTR1AHTR2ADRD3DRD4
SCHEMBL13532797 0.93 DRD2 (0.87) DRD2HTR1AHTR2ADRD3DRD4
SCHEMBL14188956 0.90 DRD2 (0.82) DRD2HTR1AHTR2ADRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 106 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112666267-B Method for detecting related substances of aripiprazole drug substance 上海上药中西制药有限公司 2023-09-26 CN claimed
CN-112666267-A Method for detecting related substances of aripiprazole medicine 上海上药中西制药有限公司 2021-04-16 CN claimed
EP-0367141-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1996-01-10 EP claimed
US-5006528-A Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-04-09 US claimed
EP-0367141-A2 Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-05-09 EP claimed
US-20260076975-A1 TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES SHANGHAI RAISING PHARMACEUTICAL CO LTD (CN) 2026-03-19 US disclosed
EP-4628098-A1 TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES Shanghai Raising Pharmaceutical Co., Ltd. (CN) 2025-10-08 EP disclosed
US-20240368115-A1 REGULATOR CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHUJING BIOPHARMA CO., LTD (CN) 2024-11-07 US disclosed
EP-4382521-A1 REGULATOR CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shujing Biopharma Co., Ltd (CN) 2024-06-12 EP disclosed
WO-2024114781-A1 TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES 上海日馨医药科技股份有限公司 2024-06-06 WO disclosed
US-20240024310-A1 CARBOSTYRIL DERIVATIVES AND MOOD STABILIZERS FOR TREATING MOOD DISORDERS OTSUKA PHARMA CO LTD (JP) 2024-01-25 US disclosed
US-20240024310-A1 CARBOSTYRIL DERIVATIVES AND MOOD STABILIZERS FOR TREATING MOOD DISORDERS OTSUKA PHARMA CO LTD (JP) 2024-01-25 US disclosed
US-20080318972-A1 5-HT1A RECEPTOR SUBTYPE AGONIST OTSUKA PHARMACEUTICAL CO., LTD. 2008-12-25 US disclosed
US-20080171752-A1 5-HT1A Receptor Subtype Agonist OTSUKA PHARMACEUTICAL CO., LTD. 2008-07-17 US disclosed
US-20080103154-A1 3, 4-dihydro-2(IH)-quinolinone and 2(1H)-quinolinone derivatives CONCERT PHARMACEUTICALS INC. (US) 2008-05-01 US disclosed
US-20080103154-A1 3, 4-dihydro-2(IH)-quinolinone and 2(1H)-quinolinone derivatives CONCERT PHARMACEUTICALS INC. (US) 2008-05-01 US disclosed
WO-2008024481-A2 3,4-DIHYDRO-2 (1H) - QUINOLINONE AND 2 (1H)-QUINOLINONE DERIVATIVES CONCERT PHARMACEUTICALS INC. (US) 2008-02-28 WO disclosed
EP-1621198-B1 Substituted carbostyril derivatives as 5-HT 1A receptor subtype agonists OTSUKA PHARMA CO LTD (JP) 2007-05-23 EP disclosed
US-20070031513-A1 Carbostyril derivatives and mood stabilizers for treating mood disorders OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-02-08 US disclosed
US-20070031513-A1 Carbostyril derivatives and mood stabilizers for treating mood disorders OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240368115-A1 REGULATOR CONTAINING TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF TPH1, TPH2, GAP43 DRD2 327/4885HTR1A 29/4885HTR2A 57/4885
US-20070031513-A1 Carbostyril derivatives and mood stabilizers for treating mood disorders CHRNA6, GABBR1, CHRNA5 DRD2 29/4885HTR1A 151/4885HTR2A 96/4885
US-20080103154-A1 3, 4-dihydro-2(IH)-quinolinone and 2(1H)-quinolinone derivatives SLC6A3, HTR2C, AQP4 DRD2 87/4885HTR1A 34/4885HTR2A 6/4885
US-20080318972-A1 5-HT1A RECEPTOR SUBTYPE AGONIST HTR1A, HTR5A, HTR2C DRD2 130/4885HTR1A 1/4885HTR2A 5/4885
US-20240024310-A1 CARBOSTYRIL DERIVATIVES AND MOOD STABILIZERS FOR TREATING MOOD DISORDERS DRD2, CHRNA6, GABRA6 DRD2 1/4885HTR1A 79/4885HTR2A 32/4885
US-20260076975-A1 TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES PDXK, NADK, HYPK DRD2 2783/4885HTR1A 607/4885HTR2A 445/4885
US-20080171752-A1 5-HT1A Receptor Subtype Agonist HTR1A, HTR5A, HTR2C DRD2 130/4885HTR1A 1/4885HTR2A 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.