SCHEMBL8635339

SCHEMBL8635339

COc1cccc(N(C)c2cc(C)c(C(=O)Cl)cc2S(C)(=O)=O)c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 0.42
MTNR1B P49286 9/20 0.42
HSD17B2 P37059 3/20 0.42
HSD17B1 P14061 2/20 0.42
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 1/20 0.37
ESR1 P03372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634267 0.87 KEAP1 (0.41) ALDH1A1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL8635879 0.87 MTNR1A (0.43) MTNR1AMTNR1BHSD17B2HSD17B1ALDH1A1
SCHEMBL8638285 0.85 PDE4B (0.41) LMNA
SCHEMBL8635012 0.85 NSD2 (0.36) ESR1
SCHEMBL8632179 0.84 SLC9A1 (0.54)
SCHEMBL8634338 0.84 ALDH1A1 (0.38) ALDH1A1LMNA
SCHEMBL8635870 0.81 KCNJ6 (0.39)
SCHEMBL8638262 0.80 HPGD (0.39) ALDH1A1LMNA
SCHEMBL8635629 0.79 FLT1 (0.36) ALDH1A1
SCHEMBL8634555 0.79 MKNK1 (0.38) CYP3A4CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed