SCHEMBL8634267

SCHEMBL8634267

COc1ccc(N(C)c2cc(C)c(C(=O)Cl)cc2S(C)(=O)=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.41
NFE2L2 Q16236 2/20 0.41
CYP2C9 P11712 1/20 0.39
TUBB4A P04350 2/20 0.39
TUBB P07437 2/20 0.39
TUBA3C P0DPH7 2/20 0.39
TUBA1B P68363 2/20 0.39
TUBA4A P68366 2/20 0.39
TUBB4B P68371 2/20 0.39
TUBB3 Q13509 2/20 0.39
TUBB2A Q13885 2/20 0.39
TUBB8 Q3ZCM7 2/20 0.39
TUBA3E Q6PEY2 2/20 0.39
TUBA1A Q71U36 2/20 0.39
TUBA1C Q9BQE3 2/20 0.39
TUBB6 Q9BUF5 2/20 0.39
TUBB2B Q9BVA1 2/20 0.39
TUBB1 Q9H4B7 2/20 0.39
KCNJ6 P48051 1/20 0.37
KCNJ5 P48544 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635339 0.87 MTNR1A (0.42) CYP2C9LMNACYP3A4CYP2C19ALDH1A1
SCHEMBL8635629 0.86 FLT1 (0.36) KCNJ6KCNJ5KCNJ3TP53RXRA
SCHEMBL8632126 0.86 TUBB4A (0.37) KEAP1NFE2L2TUBB4ATUBBTUBA3C
SCHEMBL8635192 0.85 RXRA (0.35) KCNJ6KCNJ5KCNJ3LMNAKMT2A
SCHEMBL8635012 0.85 NSD2 (0.36) RXRARXRBRXRG
SCHEMBL7764019 0.83 SLC9A1 (0.57)
SCHEMBL8635329 0.83 SLC9A1 (0.35) LMNARXRARXRBRXRGALDH1A1
SCHEMBL8633950 0.82 SIRT2 (0.35) RXRARXRBRXRGPDK1PDK2
SCHEMBL8635732 0.82 KCNJ6 (0.38) KCNJ6KCNJ3
SCHEMBL8638262 0.80 HPGD (0.39) LMNAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed