SCHEMBL8879527

SCHEMBL8879527

CCC(C)OC(=O)c1ccccc1C(=O)[O-].[Na+]

nearest known ligand 0.50

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A known ✓ P35498 1/20 0.45
SCN2A known ✓ Q99250 1/20 0.45
SCN3A known ✓ Q9NY46 1/20 0.45
GABRA1 known ✓ P14867 3/20 0.40
GABRG2 known ✓ P18507 3/20 0.40
GABRB3 known ✓ P28472 3/20 0.40
GABRA5 known ✓ P31644 3/20 0.40
GABRA3 known ✓ P34903 3/20 0.40
GABRA2 known ✓ P47869 3/20 0.40
GABRA6 known ✓ Q16445 1/20 0.40
CA2 known ✓ P00918 1/20 0.40
ALDH1A1 P00352 4/20 0.50
ADRA1A P35348 1/20 0.45
TSHR P16473 3/20 0.45
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
MAPT P10636 1/20 0.41
USP2 O75604 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6231293 0.90 ALDH1A1 (0.58) ALDH1A1ADRA1ATSHRSCN1ASCN2A
SCHEMBL20561123 0.83 ALDH1A1 (0.49) ALDH1A1ADRA1ATSHRSCN1ASCN2A
SCHEMBL8880799 0.83 ALDH1A1 (0.52) ALDH1A1ADRA1ATSHRSCN1ASCN2A
SCHEMBL2989810 0.83 ALDH1A1 (0.68) ALDH1A1ADRA1ATSHRSCN1ASCN2A
SCHEMBL8879331 0.83 NPC1 (0.53) ALDH1A1TSHRKDM4EHPGDCA2
SCHEMBL28815185 0.82 TSHR (0.70) ALDH1A1ADRA1ATSHRSCN1ASCN2A
SCHEMBL39200 0.80 LMNA (0.55) ALDH1A1ADRA1ATSHRSCN1ASCN2A
SCHEMBL15204568 0.80 ALDH1A1 (0.49) ALDH1A1ADRA1ATSHRSCN1ASCN2A
SCHEMBL13328208 0.80 SMN1; SMN2 (0.58) ALDH1A1ADRA1ATSHRSCN1ASCN2A
SCHEMBL15684530 0.79 ALDH1A1 (0.75) ALDH1A1ADRA1ATSHRSCN1ASCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1058002-C Method for treatment of mixture of hydroperoxide SUMITOMO CHEMICAL CO (JP) 2000-11-01 CN disclosed
US-5639922-A CONTACTING AROMATIC PRIMARY AND TERTIARY HYDROPEROXIDES MIXTURE OBTAINED BY OXIDATION OF ALKYLAROMATIC COMPOUNDS WITH AN ALKALI OR ALKALINE ORGANIC AROMATIC CARBOXYLIC ACID SALT, DECOMPOSING WITH ACID CATALYST FORMING ALKYL PHENOLS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-06-17 US disclosed
CN-1128754-A Method for treatment of mixture of hydroperoxide SUMITOMO CHEMICAL CO (JP) 1996-08-14 CN disclosed