SCHEMBL9372184

SCHEMBL9372184

COc1cccc2c1C(CC(=O)O)C(=O)CC2

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.42
HTR1A P08908 4/20 0.41
CYP2D6 P10635 1/20 0.41
MTNR1B P49286 5/20 0.40
MTNR1A P48039 4/20 0.40
HCRTR1 O43613 3/20 0.40
HCRTR2 O43614 3/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DRD2 P14416 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8900041 0.88 HTR1A (0.43) HTR2AHTR1ACYP2D6MTNR1BMTNR1A
SCHEMBL7935873 0.80 MTNR1A (0.43) HTR1ACYP2D6MTNR1BMTNR1AHCRTR1
SCHEMBL7926754 0.80 HTR1A (0.55) HTR2AHTR1AHCRTR1HCRTR2DRD2
SCHEMBL7238842 0.79 ALDH1A1 (0.38)
SCHEMBL7926523 0.78 HTR1A (0.53) HTR2AHTR1ADRD2
SCHEMBL7935755 0.76 HTR1A (0.52) HTR1AMTNR1BMTNR1AKDM4EHPGD
SCHEMBL9052842 0.75 DRD2 (0.45) HTR1AHCRTR1HCRTR2DRD2
SCHEMBL9035210 0.73 MTNR1A (0.41) HTR2AHTR1AMTNR1BMTNR1ASMN1; SMN2
SCHEMBL9441175 0.72 MTNR1B (0.44) HTR2AHTR1AMTNR1BMTNR1ADRD2
SCHEMBL24650780 0.71 AADAT (0.42) HTR2AHTR1AMTNR1BMTNR1ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0586525-A1 CARBOXAMIDO-(1,2N)-CARBOCYCLIC-2-AMINOTETRALIN DERIVATIVES. UPJOHN CO (US) 1994-03-16 EP disclosed
WO-1992020655-A1 CARBOXAMIDO-(1,2N)-CARBOCYCLIC-2-AMINOTETRALIN DERIVATIVES THE UPJOHN COMPANY (US) 1992-11-26 WO disclosed