SCHEMBL8917377

SCHEMBL8917377

CSc1ccc2c(ccc3c(C(F)F)nn(NS(=O)(=O)c4ccccc4)c32)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CCR2 P41597 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
KMT2A Q03164 1/20 0.30
EDNRB P24530 1/20 0.30
EDNRA P25101 1/20 0.30
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8920824 0.85 SLC40A1 (0.37) ALDH1A1NPSR1RXFP1EDNRBEDNRA
SCHEMBL8916155 0.84 HTR6 (0.36) ALDH1A1KMT2AHTR6
SCHEMBL8917696 0.80 GAA (0.39) ALDH1A1SMN1; SMN2KMT2AHTR6
SCHEMBL8918176 0.74 CCR3 (0.36) KMT2A
SCHEMBL8918255 0.74 PTGS2 (0.38)
SCHEMBL8918039 0.74 HSD17B1 (0.35) ALDH1A1SMN1; SMN2KMT2A
SCHEMBL8918357 0.73 HPGD (0.37) ALDH1A1KMT2A
SCHEMBL8916300 0.73 MEN1 (0.39) SMN1; SMN2KMT2AHTR6
SCHEMBL8917789 0.73 HTR6 (0.38) ALDH1A1SMN1; SMN2KMT2AHTR6
SCHEMBL8917165 0.72 CYP1A2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed