SCHEMBL8918560

SCHEMBL8918560

CC(=O)c1cnc2c(c1)oc(=O)n2CCc1ccncc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
IDO1 P14902 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
THRB P10828 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
ASAH1 Q13510 1/20 0.34
NPY5R Q15761 1/20 0.34
PDE1B Q01064 1/20 0.34
IMPDH2 P12268 1/20 0.34
PKM P14618 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
SLC6A2 P23975 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918738 0.90 ALDH1A1 (0.50) LMNATSHRALDH1A1MAPK1IDO1
SCHEMBL8919804 0.82 LMNA (0.42) LMNATSHRALDH1A1MAPK1IDO1
SCHEMBL8918012 0.78 MIF (0.47) LMNATSHRALDH1A1PDE1BHTT
SCHEMBL8917032 0.78 CYP1A2 (0.36) ALDH1A1MAPK1MEN1KMT2ASIGMAR1
SCHEMBL8624599 0.75 ADORA2B (0.35) ALDH1A1SIGMAR1PDE1BSLC6A2HTR2A
SCHEMBL8626905 0.75 ALDH1A1 (0.43) LMNAALDH1A1SIGMAR1PDE1BPKM
SCHEMBL8625029 0.64 NPC1 (0.48) TSHRALDH1A1HTTKDM4E
SCHEMBL8917897 0.64 SIGMAR1 (0.42) LMNAALDH1A1MAPK1SIGMAR1SMN1; SMN2
SCHEMBL8918636 0.64 HSD17B10 (0.43) LMNATSHRALDH1A1MAPK1PKM
SCHEMBL8626022 0.63 ALDH1A1 (0.63) LMNATSHRALDH1A1MAPK1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed