SCHEMBL8917032

SCHEMBL8917032

CC(=O)c1cnc2c(c1)oc(=O)n2CCC#N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 11/20 0.36
ALDH1A1 P00352 9/20 0.36
HSD17B10 Q99714 9/20 0.36
CASP1 P29466 8/20 0.36
CASP7 P55210 8/20 0.36
CYP2C9 P11712 4/20 0.36
HPGD P15428 4/20 0.36
KMO O15229 2/20 0.35
MAPK1 P28482 3/20 0.34
CYP2C19 P33261 3/20 0.34
MAPT P10636 1/20 0.34
CYP3A4 P08684 3/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
USP2 O75604 3/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8624599 0.88 ADORA2B (0.35) ALDH1A1KMOPDE4APDE4BPDE4C
SCHEMBL8918139 0.81 HSD17B10 (0.38) CYP1A2ALDH1A1HSD17B10CASP1CASP7
SCHEMBL8918738 0.79 ALDH1A1 (0.50) ALDH1A1HPGDMAPK1MAPTMEN1
SCHEMBL8918560 0.78 LMNA (0.38) ALDH1A1MAPK1MEN1KMT2ASIGMAR1
SCHEMBL8626905 0.77 ALDH1A1 (0.43) ALDH1A1HSD17B10HPGDMAPTSIGMAR1
SCHEMBL8918012 0.76 MIF (0.47) ALDH1A1HSD17B10HPGDMAPTTP53
SCHEMBL8627148 0.67 PDE4B (0.36) ALDH1A1HSD17B10HPGDKMOMAPK1
SCHEMBL8917897 0.66 SIGMAR1 (0.42) ALDH1A1HPGDMAPK1SIGMAR1GAA
SCHEMBL8625701 0.65 ALDH1A1 (0.40) ALDH1A1HSD17B10HPGDMEN1KMT2A
SCHEMBL8919469 0.63 MAPK1 (0.36) ALDH1A1HSD17B10HPGDMAPK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed