SCHEMBL8947000

SCHEMBL8947000

COc1ccc2c(N)onc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.43
ALDH1A1 P00352 4/20 0.43
CYP3A4 P08684 2/20 0.43
NCF1 P14598 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
NQO2 P16083 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HPGD P15428 2/20 0.41
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
APP P05067 1/20 0.41
CLK1 P49759 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21596926 0.86 MEN1 (0.48) ACHEALDH1A1CYP3A4NCF1MEN1
SCHEMBL21596938 0.75 LMNA (0.37) ALDH1A1LMNATP53CA2
SCHEMBL21596940 0.72 ENPP2 (0.45) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL9214142 0.72 NR4A2 (0.47) ACHEALDH1A1CYP3A4MEN1KMT2A
SCHEMBL6952286 0.71 CLK1 (0.50) ALDH1A1CYP3A4KDM4ENPC1LMNA
SCHEMBL5178348 0.71 L3MBTL1 (0.44) ALDH1A1MEN1KMT2AKDM4ENPC1
SCHEMBL8772682 0.71 ALDH1A1 (0.38) ALDH1A1MEN1KMT2AKDM4ENPC1
SCHEMBL11195844 0.70 ALDH1A1 (0.52) ACHEALDH1A1CYP3A4NCF1MEN1
SCHEMBL21596922 0.68 KMT2A (0.50) ALDH1A1CYP3A4MEN1KMT2AKDM4E
SCHEMBL3841526 0.68 HTR1A (0.58) ALDH1A1CYP3A4NCF1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5580982-A ANTIDEPRESSANTS; ANTICHOLINERGIC AGENTS; ALZHEIMER'S DISEASE; AMINE OXIDASE INHIBITORS HOECHST MARION ROUSSEL INC. (US) 1996-12-03 US disclosed