SCHEMBL8963670

SCHEMBL8963670

COc1ccc(-c2nc(C(C(c3ccccc3)c3ccccc3)N3CCNCC3)c(C)[nH]2)c(OC)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.42
SLC6A2 P23975 3/20 0.41
SLC6A4 P31645 3/20 0.41
TLR9 Q9NR96 2/20 0.39
TLR7 Q9NYK1 2/20 0.39
SLC6A3 Q01959 2/20 0.39
KCNH2 Q12809 2/20 0.39
CYP2D6 P10635 1/20 0.39
HTR7 P34969 1/20 0.39
HTR1A P08908 1/20 0.38
HTR3A P46098 1/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
TACR1 P25103 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
CRHR1 P34998 2/20 0.36
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963762 0.89 HTR7 (0.44) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL8964068 0.85 PRMT5 (0.44) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL8963561 0.85 SLC6A2 (0.47) SLC6A2SLC6A4CYP2D6HTR7HTR1A
SCHEMBL8963552 0.81 SLC6A4 (0.42) SLC6A2SLC6A4CYP2D6HTR7HTR1A
SCHEMBL8963679 0.79 MEN1 (0.42) SLC6A2SLC6A4DRD2DRD4DRD3
SCHEMBL8963956 0.79 SLC6A4 (0.40) SLC6A2SLC6A4SLC6A3CYP2D6HTR7
SCHEMBL8963532 0.78 SLC6A2 (0.41) SLC6A2SLC6A4CYP2D6HTR7HTR1A
SCHEMBL8963737 0.77 OPRM1 (0.38) TLR9TLR7HTR7HTR1AHTR3A
SCHEMBL8969991 0.77 OPRD1 (0.37) SLC6A2SLC6A4KCNH2CYP1A2TACR1
SCHEMBL8963580 0.77 PRMT5 (0.40) SLC6A2SLC6A4CYP1A2CYP3A4TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514800-A CALCIUM CHANNEL BLOCKERS, CEREBRAL ISCHEMIA SYNTEX PHARMACEUTICALS, LTD. (GB) 1996-05-07 US disclosed