Phthalimide

Phthalimide

SCHEMBL8983753

O.O=C1NC(=O)c2ccccc21.O=C1NC(=O)c2ccccc21

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Phthalimide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B known ✓ P49841 1/20 0.94
PARP1 known ✓ P09874 4/20 0.56
ACVR1 known ✓ Q04771 1/20 0.56
MEN1 known ✓ O00255 4/20 0.47
EGFR known ✓ P00533 1/20 0.46
THRB known ✓ P10828 2/20 0.45
PARP2 known ✓ Q9UGN5 1/20 0.44
CASP7 P55210 3/20 0.75
CASP3 P42574 2/20 0.75
CASP6 P55212 2/20 0.75
CASP8 Q14790 2/20 0.75
CASP2 P42575 1/20 0.75
PDGFRA P16234 1/20 0.56
FER P16591 1/20 0.56
LTK P29376 1/20 0.56
CDK8 P49336 1/20 0.56
LRRK2 Q5S007 1/20 0.56
DYRK1B Q9Y463 1/20 0.56
MAPK1 P28482 4/20 0.52
LMNA P02545 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phthalimide SCHEMBL27572997 1.00 GSK3B (0.94) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL28226707 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL7771670 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL29366030 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL64 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL11040503 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL10192661 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL30125197 0.97 GSK3B (1.00) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL28074926 0.94 GSK3B (0.83) GSK3BCASP7CASP3CASP6CASP8
Phthalimide SCHEMBL228977 0.94 GSK3B (0.94) GSK3BCASP7CASP3CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101550102-B Method for preparing di-(N-methyl phthalimide) ether UNIV NORTHWEST A&F 2010-12-01 CN claimed
CN-101139315-B Method for preparing di(N-methyl phthalimide) ether SHANGHAI RES INST SYNTHETIC RESINS 2010-04-07 CN claimed
CN-101550102-A Preparation method of bis- (N-methyl phthalimide) ether UNIV NORTHWEST A&F (CN) 2009-10-07 CN claimed
CN-100460390-C Bi(N-methylphthalic imidine) ester preparation method SHANGHAI INST TECHNOLOGY (CN) 2009-02-11 CN claimed
CN-101139315-A Method for preparing di(N-methyl phthalimide) ether SHANGHAI RES INST OF SYNTHETIC (CN) 2008-03-12 CN claimed
CN-101007782-A Bi(N-methylphthalic imidine) ester preparation method SHANGHAI INST TECHNOLOGY (CN) 2007-08-01 CN claimed
EP-0274601-A2 Synthesis of bis (n-substituted phthalimide) ethers GENERAL ELECTRIC COMPANY (US) 1988-07-20 EP claimed
US-4757149-A Synthesis of bis(N-substituted phthalimide)ethers GENERAL ELECTRIC COMPANY (US) 1988-07-12 US claimed
US-11866417-B2 Crystalline 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione hemihydrate, compositions and methods of use thereof CELGENE CORPORATION (US) 2024-01-09 US disclosed
US-20220031661-A1 SMALL MOLECULE INHIBITORS OF THE BFRB:BFD INTERACTION UNIVERSITY OF KANSAS 2022-02-03 US disclosed
WO-2020117832-A1 SMALL MOLECULE INHIBITORS OF THE BFRB:BFD INTERACTION UNIVERSITY OF KANSAS (US) 2020-06-11 WO disclosed
CN-103539931-A Preparation method of catalyst for synthesizing medium and low-molecular weight polyethylene oxide SHANGHAI LIAN SHENG CHEMICAL CO LTD 2014-01-29 CN disclosed
CN-101550102-B Method for preparing di-(N-methyl phthalimide) ether UNIV NORTHWEST A&F 2010-12-01 CN disclosed
CN-101139315-B Method for preparing di(N-methyl phthalimide) ether SHANGHAI RES INST SYNTHETIC RESINS 2010-04-07 CN disclosed
EP-0274601-A2 Synthesis of bis (n-substituted phthalimide) ethers GENERAL ELECTRIC COMPANY (US) 1988-07-20 EP disclosed
EP-0274601-A2 Synthesis of bis (n-substituted phthalimide) ethers GENERAL ELECTRIC COMPANY (US) 1988-07-20 EP disclosed
EP-0274601-A2 Synthesis of bis (n-substituted phthalimide) ethers GENERAL ELECTRIC COMPANY (US) 1988-07-20 EP disclosed
US-4757149-A Synthesis of bis(N-substituted phthalimide)ethers GENERAL ELECTRIC COMPANY (US) 1988-07-12 US disclosed
US-4757149-A Synthesis of bis(N-substituted phthalimide)ethers GENERAL ELECTRIC COMPANY (US) 1988-07-12 US disclosed
US-4757149-A Synthesis of bis(N-substituted phthalimide)ethers GENERAL ELECTRIC COMPANY (US) 1988-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11866417-B2 Crystalline 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione hemihydrate, compositions and methods of use thereof QDPR, HTR3D, IAPP GSK3B 2241/4885PARP1 2244/4885ACVR1 2830/4885
US-20220031661-A1 SMALL MOLECULE INHIBITORS OF THE BFRB:BFD INTERACTION BLVRB, TFPI, ETFB GSK3B 4352/4885PARP1 4494/4885ACVR1 4040/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.