SCHEMBL9020233

SCHEMBL9020233

CN1C2CCCC1(c1n[nH]c3ccccc13)CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
CHRNA7 P36544 5/20 0.37
HTR3A P46098 2/20 0.37
KDM4E B2RXH2 4/20 0.35
GAA P10253 2/20 0.35
PDPK1 O15530 1/20 0.35
CYP3A4 P08684 1/20 0.35
HPGD P15428 2/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CYP1A2 P05177 1/20 0.34
YTHDC1 Q96MU7 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9020428 0.83 HTR2A (0.40) HTR2A
SCHEMBL29435414 0.76 HTR6 (0.40) CHRNA7HTR3AKDM4ECYP3A4MEN1
SCHEMBL7968110 0.76 HTR6 (0.40) CHRNA7HTR3AKDM4ECYP3A4MEN1
SCHEMBL633353 0.72 SLC6A2 (0.43) SIGMAR1KCNH2
SCHEMBL7973508 0.71 HRH3 (0.38) CHRNA7KDM4EALDH1A1
SCHEMBL7121073 0.68 OPRL1 (0.35) CYP3A4MEN1KMT2AKCNH2
SCHEMBL30189641 0.68 KCNH2 (0.33) KCNH2
SCHEMBL7898112 0.67 OPRK1 (0.31)
SCHEMBL7458612 0.65 OPRM1 (0.34) KMT2A
SCHEMBL1843463 0.65 ALDH1A1 (0.34) KDM4EKCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498331-B1 N-(aryloxyalkyl)heteroaryl-8-azabicyclo(3.2.1)octanes, intermediates and a process for the preparation thereof and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-05-22 EP disclosed
US-5340936-A Antipsychotic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-08-23 US disclosed
US-5334599-A Heteroaryl-8-azabicyclo[3,2,1]octanes as antipsychotic agents, 5-HT3 receptor antagonists and inhibitors of the reuptake of serotonin HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-08-02 US disclosed
US-5234931-A Anxiolytic agents; antdepressants; schizophrenia; drug abuse; medical diagnosis HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-08-10 US disclosed
EP-0498331-A1 N-(aryloxyalkyl)heteroaryl-8-azabicyclo(3.2.1)octanes, intermediates and a process for the preparation thereof and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-08-12 EP disclosed