SCHEMBL9025946

SCHEMBL9025946

COc1ccccc1-c1ncccc1C(N)c1occ2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.40
PDE5A O76074 2/20 0.39
AURKA O14965 1/20 0.39
ALDH1A1 P00352 5/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
HPGD P15428 2/20 0.39
GPR84 Q9NQS5 1/20 0.38
ADORA1 P30542 1/20 0.37
KDM4E B2RXH2 4/20 0.36
GAA P10253 3/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
PKM P14618 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 2/20 0.35
USP2 O75604 1/20 0.34
GLA P06280 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025454 0.78 CA12 (0.34) PDE5AALDH1A1SMN1; SMN2GPR84KDM4E
SCHEMBL9025514 0.76 PDE4A (0.39) ALDH1A1SMN1; SMN2KDM4ENPC1PKM
SCHEMBL9026008 0.75 PKM (0.38) GPR84PKMSYK
SCHEMBL9026859 0.74 ADRA2A (0.45) ALDH1A1HPGDKDM4EHSD17B10NPC1
SCHEMBL9025089 0.74 KDM4E (0.41) ALDH1A1SMN1; SMN2HPGDGPR84KDM4E
SCHEMBL9025520 0.74 METAP2 (0.38) ALDH1A1HPGDGPR84KDM4EGAA
SCHEMBL9032018 0.73 DHFR (0.39) ALDH1A1SMN1; SMN2HPGDKDM4EGAA
SCHEMBL9026336 0.73 CYP11B2 (0.47) ALDH1A1SMN1; SMN2KDM4EGAAHSD17B10
SCHEMBL9024896 0.73 MYB (0.36) GPR84NPC1RAB9ALMNA
SCHEMBL9025568 0.73 METAP2 (0.39) ADORA2AALDH1A1GPR84KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed