SCHEMBL9255250

SCHEMBL9255250

Cc1cc(C)nc(NCC2=COc3cc(O)ccc3O2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.35
NOS3 P29474 1/20 0.35
NOS2 P35228 1/20 0.35
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 4/20 0.34
HSD17B10 Q99714 4/20 0.34
KDM4E B2RXH2 4/20 0.34
HPGD P15428 3/20 0.34
GAA P10253 2/20 0.34
ALOX15 P16050 2/20 0.34
CASP1 P29466 2/20 0.34
TP53 P04637 1/20 0.34
GLA P06280 1/20 0.34
CASP7 P55210 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9259716 0.75 LCK (0.45) NPC1RAB9ASMN1; SMN2KMT2AALDH1A1
SCHEMBL9255245 0.68
SCHEMBL7021029 0.65 MTNR1A (0.51) NPC1RAB9ASMN1; SMN2KMT2AALDH1A1
SCHEMBL10889658 0.65 LMNA (0.51) IDH1HSD17B10GAACHRNB2CHRNB4
SCHEMBL7157836 0.64 NPSR1 (0.50) IDH1NOS3NOS2KMT2AALDH1A1
SCHEMBL1949112 0.64 NOS3 (0.53) IDH1NOS3NOS2NPC1RAB9A
SCHEMBL2831934 0.63 NOS2 (0.48) IDH1NOS3NOS2NPC1RAB9A
SCHEMBL9258029 0.63 DRD3 (0.37) HSD17B10KDM4ECYP3A4
SCHEMBL5175721 0.62 ALPL (0.51) IDH1NOS3NOS2RAB9AKMT2A
SCHEMBL1948938 0.61 NOS3 (0.50) IDH1NOS3NOS2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5439909-A 2-Substituted with amide or thioamide group; antioxidant for lipoproteins, antilipemic agents, anticholesterol agents ADIR ET COMPAGNIE (FR) 1995-08-08 US disclosed
US-5420132-A Antilipemic agents ADIR ET COMPAGNIE (FR) 1995-05-30 US disclosed
EP-0624582-A1 Substituted benzodioxine, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-11-17 EP disclosed