Methylene Chloride

Methylene Chloride

SCHEMBL9305751

CCN(CC)CC.CO.ClCCl.O

nearest known ligand 0.32

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Methylene Chloride. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 1/20 0.31
THRB known ✓ P10828 1/20 0.31
CACNA1B known ✓ Q00975 1/20 0.31
CYP2C9 P11712 2/20 0.32
HPGD P15428 2/20 0.32
MAPK1 P28482 2/20 0.32
HSD17B10 Q99714 2/20 0.32
CYP1A2 P05177 1/20 0.32
HIF1A Q16665 1/20 0.32
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
APEX1 P27695 1/20 0.31
HTT P42858 1/20 0.31
RECQL P46063 1/20 0.31
APBA1 Q02410 1/20 0.31
KMT2A Q03164 1/20 0.31
MCL1 Q07820 1/20 0.31
HKDC1 Q2TB90 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylene Chloride SCHEMBL153756 0.96 CYP2C9 (0.33) CYP2C9HPGDMAPK1HSD17B10CYP1A2
Methyl Alcohol SCHEMBL946877 0.89 ALDH1A1 (0.35) CYP2C9HPGDMAPK1HSD17B10CYP1A2
Methylene Chloride SCHEMBL187626 0.89 ALDH1A1 (0.36) CYP2C9HPGDMAPK1HSD17B10CYP1A2
Acetonitrile SCHEMBL5210744 0.88
Methylene Chloride SCHEMBL10795300 0.86 KDM4E (0.30) MAPK1ALDH1A1KDM4EMEN1POLB
Alcohol SCHEMBL946131 0.86 ALDH1A1 (0.43) CYP2C9HPGDMAPK1HSD17B10CYP1A2
Methylene Chloride SCHEMBL15348142 0.85 ALDH1A1 (0.33) ALDH1A1
Methylene Chloride SCHEMBL14696854 0.85 LMNA (0.35) ALDH1A1MAPTHTT
Methylene Chloride SCHEMBL9555746 0.85 ALDH1A1 (0.33) ALDH1A1
Chloromethane SCHEMBL375766 0.85 CYP2C9 (0.35) CYP2C9HPGDMAPK1HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102759598-A Quality detection method for 29-componnet stagnation dissipation powder as Tibetan medicinal composition and preparations thereof SHANDONG ARURA PHARMACEUTICAL RES & DEV CO LTD 2012-10-31 CN claimed
CN-102749401-A Quality inspection method of traditional Chinese medicine composition twenty-five-ingredient lung disease preparation SHANDONG ARURA PHARMACEUTICAL RES & DEV CO LTD 2012-10-24 CN claimed
CN-115792075-B Detection method of 4' -monophosphoryl lipid A compound 江苏瑞科生物技术股份有限公司 2023-11-03 CN disclosed
CN-115792075-A Detection method of 4' -monophosphoryl lipid A compound 江苏瑞科生物技术股份有限公司 2023-03-14 CN disclosed
CN-102759598-B Quality detection method for 29-componnet stagnation dissipation powder as Tibetan medicinal composition and preparations thereof SHANDONG ARURA PHARMACEUTICAL RESEARCH & DEVELOPMENT CO., LTD. (CN) 2014-10-15 CN disclosed
CN-102749401-B Inspection method of traditional Chinese medicine composition twenty-five-ingredient lung disease preparation SHANDONG ARURA PHARMACEUTICAL RES & DEV CO LTD 2013-12-18 CN disclosed
CN-102759598-A Quality detection method for 29-componnet stagnation dissipation powder as Tibetan medicinal composition and preparations thereof SHANDONG ARURA PHARMACEUTICAL RES & DEV CO LTD 2012-10-31 CN disclosed
CN-102749401-A Quality inspection method of traditional Chinese medicine composition twenty-five-ingredient lung disease preparation SHANDONG ARURA PHARMACEUTICAL RES & DEV CO LTD 2012-10-24 CN disclosed
EP-0495265-B1 Acid-labile linker molecules AKZO NOBEL NV (NL) 1994-08-03 EP disclosed
US-5306809-A Cancer immune therapy AKZO N.V. (NL) 1994-04-26 US disclosed
US-5296597-A Antibiotics SPA SOCIETA' PRODOTTI ANTIBIOTICI S.P.A. (IT) 1994-03-22 US disclosed
EP-0495265-A1 Acid-labile linker molecules Akzo Nobel N.V. (NL) 1992-07-22 EP disclosed