3-O-Methyl-Alpha-Methyldopamine

3-O-Methyl-Alpha-Methyldopamine

SCHEMBL9434236

COc1cc(CC(C)N)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOS P01100 1/20 0.75
TTR P02766 1/20 0.75
JUN P05412 1/20 0.75
NR3C1 P04150 1/20 0.75
HSD17B1 P14061 1/20 0.75
HSD17B2 P37059 1/20 0.75
ALOX15 P16050 3/20 0.69
ALOX12 P18054 3/20 0.69
MMP1 P03956 1/20 0.66
CYP3A4 P08684 1/20 0.66
TAAR1 Q96RJ0 2/20 0.62
TSHR P16473 2/20 0.62
MAPK1 P28482 1/20 0.62
LMNA P02545 1/20 0.60
GLA P06280 1/20 0.60
GAA P10253 2/20 0.56
MAPT P10636 1/20 0.56
ATM Q13315 1/20 0.56
ALDH1A1 P00352 1/20 0.54
NFKB1 P19838 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
3-O-Methyl-Alpha-Methyldopamine SCHEMBL28514447 1.00 FOS (0.75) FOSTTRJUNNR3C1HSD17B1
3-O-Methyl-Alpha-Methyldopamine SCHEMBL9434243 1.00 FOS (0.75) FOSTTRJUNNR3C1HSD17B1
SCHEMBL28002729 0.86 ALOX15 (0.75) FOSTTRJUNNR3C1HSD17B1
Dihydroguaiaretic Acid SCHEMBL9087980 0.86 FOS (1.00) FOSTTRJUNNR3C1HSD17B1
Mesodihydroguaiaretic Acid SCHEMBL974725 0.86 FOS (1.00) FOSTTRJUNNR3C1HSD17B1
SCHEMBL11571527 0.86 FOS (0.80) FOSTTRJUNNR3C1HSD17B1
SCHEMBL10509993 0.85 FOS (0.68) FOSTTRJUNNR3C1HSD17B1
SCHEMBL19337385 0.84 FOS (0.77) FOSTTRJUNNR3C1HSD17B1
SCHEMBL14532804 0.84 FOS (0.77) FOSTTRJUNNR3C1HSD17B1
SCHEMBL2564908 0.84 LDHA (0.59) ALOX15ALOX12TAAR1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220273680-A1 Methods of Treating Psychological and Brain Disorders UNIVERSITY OF MARYLAND, BALTIMORE (US) 2022-09-01 US claimed
EP-4013403-A1 METHODS OF TREATING PSYCHOLOGICAL AND BRAIN DISORDERS University of Maryland, Baltimore (US) 2022-06-22 EP claimed
WO-2021030571-A1 METHODS OF TREATING PSYCHOLOGICAL AND BRAIN DISORDERS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2021-02-18 WO claimed
US-12590077-B2 Short-acting monoamine releasers Solvonics Therapeutics Ireland Holdings Limited (IE) 2026-03-31 US disclosed
EP-4611738-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME Lykos Therapeutics, Inc. (US) 2025-09-10 EP disclosed
US-20250134856-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME MAPS PUBLIC BENEFIT CORPORATION 2025-05-01 US disclosed
US-20250134855-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME MAPS PUBLIC BENEFIT CORPORATION 2025-05-01 US disclosed
US-20250127756-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME MAPS PUBLIC BENEFIT CORPORATION 2025-04-24 US disclosed
US-20250127757-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME MAPS PUBLIC BENEFIT CORPORATION 2025-04-24 US disclosed
US-20250100990-A1 1,3-BENZODIOXOLE ESTERS AND THEIR THERAPEUTIC USE AWAKN LS EUROPE HOLDINGS LIMITED (IE) 2025-03-27 US disclosed
WO-2024234014-A1 SUBLINGUAL SPRAY FORMULATIONS OF PSYCHEDELICS SPIRITUS BIOSCIENCE, INC. (US) 2024-11-14 WO disclosed
EP-2848617-B1 DIARYL[A, G]QUINOLIZIDINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION, AND USES THEREOF SHANGHAI INST MATERIA MEDICA CAS (CN) 2022-01-12 EP disclosed
WO-2021030571-A1 METHODS OF TREATING PSYCHOLOGICAL AND BRAIN DISORDERS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2021-02-18 WO disclosed
US-10000555-B2 Monomethylvaline compounds having phenylalanine side-chain modification at the C-terminus SEATTLE GENETICS, INC. (US) 2018-06-19 US disclosed
US-9751882-B2 Diaryl[A, G]quinolizidine compound, preparation method therefor, pharmaceutical composition, and uses thereof KINGSOUND & PARTNER (CN) 2017-09-05 US disclosed
US-20150141419-A1 DIARYL[A, G]QUINOLIZIDINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION, AND USES THEREOF SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2015-05-21 US disclosed
EP-2848617-A1 DIARYL[A, G]QUINOLIZIDINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION, AND USES THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2015-03-18 EP disclosed
US-20130123465-A1 MONOMETHYLVALINE COMPOUNDS HAVING PHENYLALANINE SIDE-CHAIN MODIFICATIONS AT THE C-TERMINUS SEATTLE GENETICS, INC. (US) 2013-05-16 US disclosed
US-8343928-B2 Monomethylvaline compounds having phenylalanine side-chain replacements at the C-terminus SEATTLE GENETICS, INC. (US) 2013-01-01 US disclosed
WO-1994000432-A1 ANORECTIC EPINEPHRINE DERIVATIVES THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1994-01-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250100990-A1 1,3-BENZODIOXOLE ESTERS AND THEIR THERAPEUTIC USE DBH, TSPO, DDO FOS 3431/4885TTR 3829/4885JUN 3572/4885
US-20250127756-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME SLC6A3, SLC6A2, SLC18A1 FOS 4195/4885TTR 855/4885JUN 4788/4885
US-20130123465-A1 MONOMETHYLVALINE COMPOUNDS HAVING PHENYLALANINE SIDE-CHAIN MODIFICATIONS AT THE C-TERMINUS MMAB, PTMS, DNPEP FOS 3009/4885TTR 3468/4885JUN 4301/4885
US-12590077-B2 Short-acting monoamine releasers SLC6A2, NPY2R, SLC6A3 FOS 4253/4885TTR 3508/4885JUN 3872/4885
US-20150141419-A1 DIARYL[A, G]QUINOLIZIDINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION, AND USES THEREOF HTR5A, HTR1F, QDPR FOS 3347/4885TTR 2670/4885JUN 4386/4885
US-20250127757-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME SLC6A3, SLC6A2, SLC18A1 FOS 4195/4885TTR 855/4885JUN 4788/4885
US-20250134856-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME SLC6A3, SLC6A2, SLC18A1 FOS 4195/4885TTR 855/4885JUN 4788/4885
US-20250134855-A1 COMPOSITIONS COMPRISING MDMA AND METHODS OF USING SAME SLC6A3, SLC6A2, SLC18A1 FOS 4195/4885TTR 855/4885JUN 4788/4885
US-10000555-B2 Monomethylvaline compounds having phenylalanine side-chain modification at the C-terminus PTMS, MMAB, DNPEP FOS 2951/4885TTR 3584/4885JUN 4310/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.