SCHEMBL9503470

SCHEMBL9503470

CCCC(NC(C)=O)(Oc1c(OC)cccc1OC)C1CCCc2c1ccc(OCc1ccccc1)c2OCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ACHE P22303 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
PKM P14618 1/20 0.39
AGTR2 P50052 5/20 0.38
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
KDM4E B2RXH2 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SCN9A Q15858 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
AGTR1 P30556 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9504633 0.92 PTGER4 (0.37) CA1CA2ACHENPC1RAB9A
SCHEMBL9503495 0.84 TAS1R3 (0.43) CA1CA2MTNR1AMTNR1BKDM4E
SCHEMBL9507066 0.73 TAS1R3 (0.35) ALDH1A1
SCHEMBL9503481 0.72 AGTR2 (0.40) CA1CA2ACHEAGTR2SCN9A
SCHEMBL9503474 0.71 NPC1 (0.40) CA1CA2ACHENPC1RAB9A
SCHEMBL9504551 0.70 NPSR1 (0.42)
SCHEMBL21091908 0.69 KMT2A (0.51) KDM1AMAOAMAOBL3MBTL1MEN1
SCHEMBL21091907 0.69 KMT2A (0.51) KDM1AMAOAMAOBL3MBTL1MEN1
SCHEMBL9814112 0.68 MAOA (0.45) CA1CA2ACHEAGTR2KDM1A
SCHEMBL8548581 0.67 CA1 (0.47) CA1CA2ACHEAGTR2MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0321968-B1 COMPOUNDS ACTIVE ON THE CARDIOVASCULAR SYSTEM ZAMBON GROUP S.p.A. (IT) 1993-07-28 EP disclosed
US-5151414-A Hypotensive agents SIMES SOCIETA ITALIANA MEDICINALI E SINTETICI S.P.A. (IT) 1992-09-29 US disclosed
US-5070106-A HYPOTENSIVES, CEREBRAL DISORDERS SIMES SOCIETA ITALIANA MEDICINALI E SINTETICI S.P.A. (IT) 1991-12-03 US disclosed