SCHEMBL9503474

SCHEMBL9503474

CCCC(Oc1c(OC)cccc1OC)C(=O)NCC1CCCc2c1ccc(OCc1ccccc1)c2OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
PKM P14618 1/20 0.40
RAB9A P51151 1/20 0.40
KDM4C Q9H3R0 3/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ACHE P22303 1/20 0.39
SIGMAR1 Q99720 2/20 0.38
AGTR2 P50052 4/20 0.37
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
KDM4E B2RXH2 1/20 0.37
AGTR1 P30556 2/20 0.36
KDM6B O15054 1/20 0.36
KDM1A O60341 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9504636 0.92 TAOK1 (0.38) NPC1PKMRAB9AKDM4CKDM6B
SCHEMBL9503507 0.83 TAS1R3 (0.43) KDM4CCA1CA2MTNR1AMTNR1B
SCHEMBL9504551 0.74 NPSR1 (0.42) SIGMAR1
SCHEMBL9503481 0.74 AGTR2 (0.40) CA1CA2ACHEAGTR2AGTR1
SCHEMBL9507069 0.73 ADRA2A (0.41) KDM4C
SCHEMBL9503470 0.71 CA1 (0.40) NPC1PKMRAB9ACA1CA2
SCHEMBL21091908 0.67 KMT2A (0.51) KDM1AMAOAMAOB
SCHEMBL21091907 0.67 KMT2A (0.51) KDM1AMAOAMAOB
SCHEMBL9814112 0.67 MAOA (0.45) CA1CA2ACHESIGMAR1AGTR2
SCHEMBL9504418 0.66 HTR6 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0321968-B1 COMPOUNDS ACTIVE ON THE CARDIOVASCULAR SYSTEM ZAMBON GROUP S.p.A. (IT) 1993-07-28 EP disclosed
US-5151414-A Hypotensive agents SIMES SOCIETA ITALIANA MEDICINALI E SINTETICI S.P.A. (IT) 1992-09-29 US disclosed
US-5070106-A HYPOTENSIVES, CEREBRAL DISORDERS SIMES SOCIETA ITALIANA MEDICINALI E SINTETICI S.P.A. (IT) 1991-12-03 US disclosed