SCHEMBL9727307

SCHEMBL9727307

C=CCc1cc2c(cc1OCc1ccccc1)C(C)(C)C(CC=O)O2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.36
ALDH1A1 P00352 4/20 0.36
MAPT P10636 3/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NR3C1 P04150 1/20 0.36
AKR1B1 P15121 1/20 0.35
PTPN1 P18031 1/20 0.34
KDM4E B2RXH2 3/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.33
SIRT1 Q96EB6 1/20 0.32
MAOB P27338 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727686 0.86 NR3C1 (0.38) L3MBTL1ALDH1A1MAPTGAAHPGD
SCHEMBL9727762 0.82 NR3C1 (0.38) L3MBTL1ALDH1A1MAPTGAAHPGD
SCHEMBL9727725 0.81 AKR1B1 (0.32) L3MBTL1ALDH1A1MAPTGAAHPGD
SCHEMBL14552348 0.71 MAOB (0.54) L3MBTL1ALDH1A1MAPTGAAHPGD
SCHEMBL8890308 0.69 CCNB2 (0.40) L3MBTL1MAPTGAATDP1PTPN1
SCHEMBL9727777 0.67 AKR1B1 (0.35) ALDH1A1GAAAKR1B1KDM4ELMNA
SCHEMBL5883140 0.66 MAOA (0.55) L3MBTL1ALDH1A1MAPTGAAHPGD
SCHEMBL9727633 0.65 LTA4H (0.38) ALDH1A1NR3C1AKR1B1PTGER1PTGER4
SCHEMBL9727331 0.65 MTNR1A (0.37) AKR1B1MAOBPTGER1PTGER4PTGER3
SCHEMBL9727700 0.65 MTNR1A (0.35) L3MBTL1MAPTTDP1AKR1B1PTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed