SCHEMBL9727725

SCHEMBL9727725

C=CCc1cc2c(cc1OCc1ccccc1)C(C)(C)C(CCc1ccc(SC)cc1)O2

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.32
NR3C1 P04150 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
GCK P35557 2/20 0.31
ABCB1 P08183 1/20 0.30
HTR1A P08908 1/20 0.30
DRD2 P14416 1/20 0.30
BCHE P06276 1/20 0.30
PTGER1 P34995 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727777 0.88 AKR1B1 (0.35) AKR1B1ALDH1A1GAASIRT2GCK
SCHEMBL9727686 0.84 NR3C1 (0.38) AKR1B1NR3C1ALDH1A1GAAMAPT
SCHEMBL9727307 0.81 L3MBTL1 (0.36) AKR1B1NR3C1ALDH1A1GAAMAPT
SCHEMBL9727762 0.77 NR3C1 (0.38) AKR1B1NR3C1ALDH1A1GAAMAPT
SCHEMBL9727464 0.74 KDM4E (0.36) AKR1B1ALDH1A1TDP1L3MBTL1BCHE
SCHEMBL9727660 0.70 CGAS (0.31) MAPT
SCHEMBL14552348 0.66 MAOB (0.54) ALDH1A1GAAMAPTHPGDTDP1
SCHEMBL9727633 0.63 LTA4H (0.38) AKR1B1NR3C1ALDH1A1ABCB1HTR1A
SCHEMBL9727331 0.63 MTNR1A (0.37) AKR1B1ABCB1HTR1ADRD2PTGER1
SCHEMBL9727700 0.63 MTNR1A (0.35) AKR1B1MAPTTDP1L3MBTL1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed