SCHEMBL9833135

SCHEMBL9833135

COc1cc(CCCCCCCCCCCCCCC(=O)Cc2c[nH]nc2N)cc(OC)c1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.40
CNR2 P34972 8/20 0.40
HDAC1 Q13547 2/20 0.39
HDAC6 Q9UBN7 1/20 0.39
GLS O94925 1/20 0.38
PTGS2 P35354 1/20 0.36
CYP19A1 P11511 1/20 0.36
DHODH Q02127 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837576 0.88 ALOX5 (0.46)
SCHEMBL9833350 0.86 TUBB4A (0.41) CYP19A1
SCHEMBL9834740 0.83 ALOX5 (0.44) GLSCYP19A1
SCHEMBL9832110 0.81 TDP1 (0.41) GLS
SCHEMBL9834514 0.80 HRH1 (0.41)
SCHEMBL9833469 0.80 HDAC1 (0.46) HDAC1HDAC6GLS
SCHEMBL9833181 0.79 HDAC3 (0.44) HDAC1HDAC6
SCHEMBL9832892 0.79 NAAA (0.37) GLS
SCHEMBL9833192 0.72 ALDH1A1 (0.37) HDAC1HDAC6GLS
SCHEMBL5275656 0.71 CNR1 (0.53) CNR1CNR2HDAC1HDAC6PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129846-B1 (3-AMINO-1H-PYRAZOL-4-YL)(ARYL)METHANONES AMERICAN CYANAMID COMPANY (US) 1991-05-08 EP claimed