SCHEMBL9953534

SCHEMBL9953534

Cc1cccc(-n2c(Cl)nc3ccc(I)cc3c2=O)c1F

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 2/20 0.43
PDE4D Q08499 1/20 0.42
TDO2 P48775 1/20 0.40
IDO2 Q6ZQW0 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TP53 P04637 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954119 0.84 HCAR1 (0.52) HCAR1TDO2IDO2LMNAL3MBTL1
SCHEMBL9954005 0.84 HCAR1 (0.40) HCAR1PDE4DALDH1A1LMNAL3MBTL1
SCHEMBL9952718 0.82 TDO2 (0.48) TDO2IDO2ALDH1A1L3MBTL1MEN1
SCHEMBL9954224 0.81 CDK9 (0.38) HCAR1PDE4DTDO2IDO2ALDH1A1
SCHEMBL9952976 0.81 LMNA (0.45) HCAR1TDO2IDO2ALDH1A1LMNA
SCHEMBL9955332 0.80 HCAR1 (0.51) HCAR1TDO2IDO2ALDH1A1LMNA
SCHEMBL9953501 0.80 HPD (0.47) HCAR1TDO2IDO2ALDH1A1L3MBTL1
SCHEMBL9954657 0.80 HPD (0.44) HCAR1TDO2IDO2POLB
SCHEMBL9954234 0.80 ALDH1A1 (0.53) HCAR1TDO2IDO2ALDH1A1TP53
SCHEMBL9954749 0.79 PDE7A (0.45) HCAR1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed