Lofendazam

Lofendazam

SCHEMBL1003371

O=C1CCNc2ccc(Cl)cc2N1c1ccccc1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.51
PDE4D Q08499 1/20 0.51
CHRM1 P11229 2/20 0.46
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
KMT2A Q03164 7/20 0.40
MEN1 O00255 6/20 0.40
AVPR1A P37288 2/20 0.39
HPGD P15428 2/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
HTT P42858 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
USP2 O75604 1/20 0.38
F7 P08709 1/20 0.37
PARP1 P09874 1/20 0.37
F3 P13726 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11428236 0.92 LMNA (0.43) OPRK1PDE4DCHRM1DRD2DRD4
SCHEMBL11433565 0.89 OPRK1 (0.51) OPRK1PDE4DCHRM1DRD2DRD4
SCHEMBL11435120 0.86 OPRK1 (0.40) OPRK1PDE4DCHRM1KMT2AAVPR1A
SCHEMBL11428247 0.86 KMT2A (0.38) OPRK1PDE4DCHRM1DRD2DRD4
SCHEMBL11420364 0.86 L3MBTL1 (0.54) OPRK1PDE4DKMT2AMEN1AVPR1A
SCHEMBL11419566 0.85 CNR1 (0.43) DRD2DRD4DRD3KMT2AMEN1
SCHEMBL11434613 0.84 ALDH1A1 (0.45) OPRK1PDE4DCHRM1DRD2DRD4
SCHEMBL11423308 0.84 MAPT (0.46) OPRK1PDE4DKMT2AMEN1ALDH1A1
SCHEMBL11428231 0.83 MEN1 (0.47) OPRK1PDE4DDRD2DRD4DRD3
SCHEMBL11429879 0.83 POLB (0.51) KMT2AMEN1ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 84 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-4239684-A 1,5'-Benzodiazepine-2-ones, pharmaceutical compositions thereof and method of use thereof KNOLL AG (DE) 1980-12-16 US claimed
US-20260137765-A1 METHODS OF PRODUCING SHIGA TOXIN B-SUBUNIT (STXB) MONOMERS AND OLIGOMERS, AND USES THEREOF INSTITUT CURIE (FR) 2026-05-21 US disclosed
US-12528794-B2 MAO-B inhibitor DRG-MAOB-1 for use in treatment of neurodegenerative diseases BAHCESEHIR UNIVERSITESI (TR) 2026-01-20 US disclosed
US-12527854-B2 Methods of producing Shiga toxin B-subunit (STxB) monomers and oligomers, and uses thereof INSTITUT CURIE (FR) 2026-01-20 US disclosed
US-12478613-B2 Selective MAO-B inhibitor DRG-MAOB-2 for use in treatment of neurodegenerative diseases BAHCESEHIR UNIVERSITESI (TR) 2025-11-25 US disclosed
US-20250281535-A1 ANTI-HUMAN CD45RC BINDING DOMAINS AND USES THEREOF ABOLERIS PHARMA (FR) 2025-09-11 US disclosed
EP-4401842-B1 ANTI-HUMAN CD45RC BINDING DOMAINS AND USES THEREOF ABOLERIS PHARMA (FR) 2025-08-27 EP disclosed
US-20020102215-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 US disclosed
US-6331289-B1 ULTRASOUND CONTRAST AGENTS, SUSPENSION IN AQUEOUS CARRIER LIQUID OF A REPORTER COMPRISING GAS-CONTAINING OR GAS-GENERATING MATERIAL, AGENT CAPABLE OF FORMING AT LEAST TWO TYPES OF BINDING PAIRS WITH TARGET; REPORTER BEING CONJUGATED NYCOMED IMAGING AS (NO) 2001-12-18 US disclosed
US-6264917-B1 MIXTURE OF GAS FILLED MICROBUBBLES AND RELEASING AGENT NYCOMED IMAGING AS (NO) 2001-07-24 US disclosed
US-6261537-B1 TARGETS AND ULTRASOUND DIAGNOSIS OF ACTIVE MATERIALS, AQUEOUS CARRIER LIQUIDS, CARRIERS AND FILM FORMING SURFACTANT PHOSPHATIDES NYCOMED IMAGING AS (NO) 2001-07-17 US disclosed
US-4239684-A 1,5'-Benzodiazepine-2-ones, pharmaceutical compositions thereof and method of use thereof KNOLL AG (DE) 1980-12-16 US disclosed
US-RE30293-E Process for preparing 1,5-benzodiazepine-2-ones KNOLL A.G. (DE) 1980-06-03 US disclosed
US-4108852-A Process for preparing 1,5-benzodiazepine-2-ones KNOLL AG. (DE) 1978-08-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12527854-B2 Methods of producing Shiga toxin B-subunit (STxB) monomers and oligomers, and uses thereof STXBP1, RNGTT, UPF1 OPRK1 3689/4885PDE4D 4410/4885CHRM1 2601/4885
US-12528794-B2 MAO-B inhibitor DRG-MAOB-1 for use in treatment of neurodegenerative diseases MAOB, MAOA, ME3 OPRK1 13/4885PDE4D 1980/4885CHRM1 373/4885
US-20260137765-A1 METHODS OF PRODUCING SHIGA TOXIN B-SUBUNIT (STXB) MONOMERS AND OLIGOMERS, AND USES THEREOF STXBP1, HBB, UPF1 OPRK1 3285/4885PDE4D 4257/4885CHRM1 3013/4885
US-12478613-B2 Selective MAO-B inhibitor DRG-MAOB-2 for use in treatment of neurodegenerative diseases MAOB, MAOA, HTR2B OPRK1 7/4885PDE4D 1446/4885CHRM1 994/4885
US-20020102215-A1 Diagnostic/therapeutic agents BID, FUS, FABP1 OPRK1 4110/4885PDE4D 3004/4885CHRM1 4583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.