SCHEMBL10073373

SCHEMBL10073373

Cc1cc(N)cc(C)c1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
TSHR P16473 4/20 0.43
PDE10A Q9Y233 1/20 0.37
CASP1 P29466 2/20 0.35
CYP3A4 P08684 3/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
GFER P55789 1/20 0.33
MAPK1 P28482 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
TP53 P04637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
BCL2 P10415 1/20 0.32
BCL2L1 Q07817 1/20 0.32
MCL1 Q07820 1/20 0.32
BCL2L2 Q92843 1/20 0.32
LMNA P02545 2/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23206105 0.84 ALDH1A1 (0.35) ALDH1A1TSHRPDE10ABCL2BCL2L1
SCHEMBL25860123 0.80 ALDH1A1 (0.32) ALDH1A1TSHR
SCHEMBL19625177 0.77 CA1 (0.43) ALDH1A1TSHRCYP3A4TP53TDP1
SCHEMBL5163137 0.77 RAPGEF4 (0.41) ALDH1A1TSHRGAANOS3NOS1
SCHEMBL11098641 0.76 TSHR (0.53) ALDH1A1TSHRCYP3A4GAAMAPK1
SCHEMBL22946251 0.74 LMNA (0.42) ALDH1A1GAABCL2BCL2L1MCL1
SCHEMBL807533 0.72 CYP3A4 (0.52) ALDH1A1TSHRCASP1CYP3A4POLB
Hydrogen Peroxide SCHEMBL10882706 0.72 LDHA (0.39) ALDH1A1GAATP53TDP1BCL2
SCHEMBL10073285 0.72 GABRA1 (0.42) ALDH1A1BCL2BCL2L1MCL1BCL2L2
SCHEMBL10073282 0.72 BCL2 (0.32) BCL2BCL2L1MCL1BCL2L2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230119573-A1 GAS SEPARATION MEMBRANE, GAS SEPARATION MODULE, GAS SEPARATION APPARATUS, AND POLYIMIDE COMPOUND FUJIFILM CORPORATION (JP) 2023-04-20 US disclosed
US-20210332020-A1 PHENYLSULFONYLUREA DERIVATIVES USEFUL AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-10-28 US disclosed
US-9951046-B2 TRPA1 modulators ALGOMEDIX, INC. (US) 2018-04-24 US disclosed
US-9603838-B2 RORgammaT inhibitors MERCK SHARP & DOHME CORP. (US) 2017-03-28 US disclosed
US-8114879-B2 4-piperazine-4-piperidine-1-ketone derivatives; graft v. host disease, arthritis, rheumatoid arthritis, inflammatory bowel disease, atopic dermatitis, psoriasis, asthma, allergies or multiple sclerosis; human immunodeficiency viricides SCHERING CORPORATION (US) 2012-02-14 US disclosed
US-7825121-B2 Piperazine derivatives useful as CCR5 antagonists SCHERING CORPORATION (US) 2010-11-02 US disclosed
US-7825121-B2 Piperazine derivatives useful as CCR5 antagonists SCHERING CORPORATION (US) 2010-11-02 US disclosed
US-20080188485-A1 PIPERIDINE DERIVATIVES USEFUL AS CCR5 ANTAGONISTS SCHERING CORPORATION 2008-08-07 US disclosed
US-7384944-B2 Piperazine derivatives useful as CCR5 antagonists SCHERING CORPORATION (US) 2008-06-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188485-A1 PIPERIDINE DERIVATIVES USEFUL AS CCR5 ANTAGONISTS CCR5, CXCR3, CCR2 ALDH1A1 2736/4885TSHR 504/4885PDE10A 3159/4885
US-20210332020-A1 PHENYLSULFONYLUREA DERIVATIVES USEFUL AS NLRP3 INHIBITORS NLRP3, NOD1, PYCARD ALDH1A1 3451/4885TSHR 4753/4885PDE10A 3075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.