SCHEMBL10238

SCHEMBL10238

Brc1cnc2ccccn12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.50
FLT3 P36888 2/20 0.49
ADORA3 P0DMS8 1/20 0.47
NPC1 O15118 4/20 0.45
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 2/20 0.45
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MIF P14174 1/20 0.45
PKM P14618 1/20 0.44
RAB9A P51151 3/20 0.42
GGPS1 O95749 1/20 0.41
FDPS P14324 1/20 0.41
DYRK1A Q13627 1/20 0.41
MAPK1 P28482 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21273200 0.76 ADORA3 (0.50) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL3313454 0.74 MIF (0.53) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL13325708 0.74 NPC1 (0.50) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL729145 0.74 NPSR1 (0.50) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL84864 0.74 NPSR1 (0.50) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL23132987 0.74 NPSR1 (0.53) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL20019155 0.74 NPSR1 (0.50) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL335455 0.74 PKM (0.51) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL504102 0.74 NPSR1 (0.50) NPSR1FLT3ADORA3NPC1KDM4E
SCHEMBL19748929 0.74 FLT3 (0.58) NPSR1FLT3ADORA3NPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 278 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114989167-B 3,6-dibromo or 3-bromoimidazo [1,2-a ] pyridine derivative and synthesis method thereof 江苏师范大学 2023-08-22 CN claimed
CN-114989167-A 3,6-dibromo or 3-bromo imidazo [1,2-a ] pyridine derivative and synthesis method thereof 江苏师范大学 2022-09-02 CN claimed
EP-4027995-B1 HPK1 ANTAGONISTS AND USES THEREOF NIMBUS SATURN INC (US) 2026-05-27 EP disclosed
EP-4741392-A1 1H-PYRAZOLO[4,3-C]PYRIDINE COMPOUND, AND COMPOSITION THEREOF AND USE THEREOF Shenzhen TargetRx Co., Ltd. (CN) 2026-05-13 EP disclosed
US-20260085073-A1 PYRAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY HOTSPOT THERAPEUTICS INC (US) 2026-03-26 US disclosed
US-12503477-B2 Colony stimulating factor-1 receptor (CSF-1R) inhibitors GENZYME CORPORATION 2025-12-23 US disclosed
US-20250361232-A1 SUBSTITUTED ACETYLENIC PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS KINASE INHIBITORS TAKEDA PHARMACEUTICALS USA INC (US) 2025-11-27 US disclosed
US-12258340-B2 Pyrazole MAGL inhibitors H. LUNDBECK A/S (DK) 2025-03-25 US disclosed
CN-116473965-B Pyrazole MAGL inhibitors H.隆德贝克有限公司 2025-03-18 CN disclosed
US-20250066318-A1 HETEROCYCLIC COMPOUNDS AS DYRK1A INHIBITORS PROTHENA BIOSCIENCES INC 2025-02-27 US disclosed
US-12215105-B2 HPK1 antagonists and uses thereof Nimbus Saturn, Inc. (US) 2025-02-04 US disclosed
US-20060205797-A1 Compounds for the treatment of inflammatory disorders SCHERING CORPORATION 2006-09-14 US disclosed
WO-2006019768-A1 HYDANTOIN DERIVATIVES FOR THE TREATMENT OF INFLAMMATORY DISORDERS SCHERING CORPORATION (US) 2006-02-23 WO disclosed
US-20060014750-A1 Pharmaceutical compositions for the treatment of CNS and other disorders PFIZER INC 2006-01-19 US disclosed
EP-1539733-A2 AZABICYCLIC COMPOUNDS ARE CENTRAL NERVOUS SYSTEM ACTIVE AGENTS Abbott Laboratories (US) 2005-06-15 EP disclosed
US-20040152724-A1 Azabicyclic compounds are central nervous system active agents ABBVIE INC. 2004-08-05 US disclosed
US-20040044029-A1 Azabicyclic compounds are central nervous system active agents ABBOTT LABORATORIES 2004-03-04 US disclosed
WO-2004016604-A2 AZABICYCLIC COMPOUNDS ARE CENTRAL NERVOUS SYSTEM ACTIVE AGENTS ABBOTT LABORATORIES (US) 2004-02-26 WO disclosed
US-20020177591-A1 Pharmaceutical compositions for the treatment of CNS and other discorders PFIZER INC. 2002-11-28 US disclosed
EP-1231212-A1 Pharmaceutical compositions for the treatment of disorders of the CNS and other disorders Pfizer Products Inc. (US) 2002-08-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250066318-A1 HETEROCYCLIC COMPOUNDS AS DYRK1A INHIBITORS DYRK1A, DYRK2, DYRK1B NPSR1 907/4885FLT3 582/4885ADORA3 1907/4885
US-20040152724-A1 Azabicyclic compounds are central nervous system active agents ACHE, CHRNA6, CHRNA2 NPSR1 517/4885FLT3 4212/4885ADORA3 395/4885
US-20040044029-A1 Azabicyclic compounds are central nervous system active agents ACHE, CHRNA6, CHRNA2 NPSR1 517/4885FLT3 4212/4885ADORA3 395/4885
US-20060205797-A1 Compounds for the treatment of inflammatory disorders TNF, MMP12, MMP8 NPSR1 660/4885FLT3 1924/4885ADORA3 3783/4885
US-20020177591-A1 Pharmaceutical compositions for the treatment of CNS and other discorders CHRNA7, CHRNA5, CHRNA10 NPSR1 113/4885FLT3 2096/4885ADORA3 20/4885
US-20060014750-A1 Pharmaceutical compositions for the treatment of CNS and other disorders CHRNA7, CHRNA10, CHRNA5 NPSR1 116/4885FLT3 2043/4885ADORA3 34/4885
US-12258340-B2 Pyrazole MAGL inhibitors MGLL, PNLIP, LPL NPSR1 4063/4885FLT3 1669/4885ADORA3 2943/4885
US-12503477-B2 Colony stimulating factor-1 receptor (CSF-1R) inhibitors CSF1R, CSF3R, IL1RN NPSR1 187/4885FLT3 7/4885ADORA3 1748/4885
US-20260085073-A1 PYRAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY MALT1, BCL6, BCL3 NPSR1 4146/4885FLT3 3874/4885ADORA3 4507/4885
US-20250361232-A1 SUBSTITUTED ACETYLENIC PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS KINASE INHIBITORS MAP4K2, MAP3K19, MAP3K1 NPSR1 3543/4885FLT3 148/4885ADORA3 1376/4885
US-12215105-B2 HPK1 antagonists and uses thereof PDXK, HIPK1, PCK1 NPSR1 2913/4885FLT3 2057/4885ADORA3 3903/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.