SCHEMBL1126618

SCHEMBL1126618

COCCc1c(-c2cccc(Cl)c2)c[nH]c1C(=O)C(=O)Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.40
TP53 P04637 1/20 0.39
SRC P12931 1/20 0.37
MAPK1 P28482 3/20 0.36
MAPK10 P53779 2/20 0.36
SLC6A3 Q01959 4/20 0.36
HPGD P15428 2/20 0.36
SLC6A2 P23975 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
NR3C2 P08235 1/20 0.35
AR P10275 1/20 0.35
NUDT1 P36639 2/20 0.35
SLC6A9 P48067 1/20 0.35
PDE4D Q08499 1/20 0.35
RORC P51449 1/20 0.34
RORB Q92753 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1126583 0.84 JAK2 (0.48) EGFRTP53MAPK1HPGDCYP1A2
SCHEMBL1127138 0.69 PYGL (0.34) TP53CYP1A2
SCHEMBL1126989 0.69 ALDH1A1 (0.39) EGFRTP53HPGDCYP1A2SLC6A9
SCHEMBL1127129 0.69 NUDT1 (0.42) EGFRTP53HPGDNUDT1SLC6A9
SCHEMBL1126847 0.68 MCL1 (0.37) MAPK1HPGD
SCHEMBL1989510 0.68 CNR1 (0.41) TP53MAPK1SLC6A3HPGDCYP1A2
SCHEMBL1127376 0.67 LMNA (0.40) TP53HPGDCYP1A2CYP2C19
SCHEMBL1127247 0.62 HTT (0.48) MAPK1HPGDSTK3
SCHEMBL1127700 0.62 KDM4E (0.40) HPGD
SCHEMBL10508590 0.62 SLC6A3 (0.54) EGFRSLC6A3HPGDSLC6A2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed