Water

Water

SCHEMBL1176982

CCCCc1nccn1C.O

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FDPS known ✓ P14324 1/20 0.41
MEN1 known ✓ O00255 2/20 0.40
AGTR1 known ✓ P30556 1/20 0.36
DRD4 known ✓ P21917 1/20 0.35
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
TLR8 Q9NR97 2/20 0.42
KCNH2 Q12809 3/20 0.39
LPO P22079 1/20 0.39
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
AGTR2 P50052 1/20 0.36
HTT P42858 1/20 0.36
APLNR P35414 1/20 0.35
TLR7 Q9NYK1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL40842 0.98 KMT2A (0.46) KMT2AALDH1A1POLBTLR8FDPS
Hydrochloric Acid SCHEMBL28330230 0.96 KMT2A (0.44) KMT2AALDH1A1POLBTLR8FDPS
Hydrochloric Acid SCHEMBL204294 0.96 TLR8 (0.44) KMT2AALDH1A1POLBTLR8FDPS
Fluoride SCHEMBL15156374 0.96 KMT2A (0.44) KMT2AALDH1A1POLBTLR8FDPS
Iodide SCHEMBL526909 0.96 KMT2A (0.44) KMT2AALDH1A1POLBTLR8FDPS
Methane SCHEMBL28225457 0.96 KMT2A (0.44) KMT2AALDH1A1POLBTLR8FDPS
Hydrochloric Acid SCHEMBL28021855 0.96 KMT2A (0.44) KMT2AALDH1A1POLBTLR8FDPS
Bromide SCHEMBL15532009 0.96 KMT2A (0.44) KMT2AALDH1A1POLBTLR8FDPS
Bromide SCHEMBL204550 0.96 KMT2A (0.44) KMT2AALDH1A1POLBTLR8FDPS
Bromide SCHEMBL28281143 0.94 KMT2A (0.43) KMT2AALDH1A1POLBTLR8FDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111560005-B Preparation method of 2-thiopheneacetyl chloride 安达市海纳贝尔化工有限公司 2022-02-18 CN claimed
CN-111560005-A Preparation method of 2-thiopheneacetyl chloride 安达市海纳贝尔化工有限公司 2020-08-21 CN claimed
CN-109796627-A A kind of stable type phosphate plasticizer and preparation method thereof 天津利海石化有限公司 2019-05-24 CN claimed
CN-109134377-A A kind of preparation method of ionic liquid 郑州工程技术学院 2019-01-04 CN claimed
CN-111560005-B Preparation method of 2-thiopheneacetyl chloride 安达市海纳贝尔化工有限公司 2022-02-18 CN disclosed
CN-111560005-A Preparation method of 2-thiopheneacetyl chloride 安达市海纳贝尔化工有限公司 2020-08-21 CN disclosed
CN-109134377-A A kind of preparation method of ionic liquid 郑州工程技术学院 2019-01-04 CN disclosed
CN-101489993-B Method for producing polyfunctional compound NITTO DENKO CORP 2013-11-06 CN disclosed
US-8168764-B2 Polyfunctional compound, optical recording material, optical recording medium, optical recording/reproducing apparatus, optical waveguide material, and photo-alignment film material NITTO DENKO CORPORATION (JP) 2012-05-01 US disclosed
US-8158737-B2 Method for production of polyfunctional compound NITTO DENKO CORPORATION (JP) 2012-04-17 US disclosed
US-8158736-B2 Method for production of polyfunctional compound NITTO DENKO CORPORATION (JP) 2012-04-17 US disclosed
US-20110098454-A1 METHOD FOR PRODUCTION OF POLYFUNCTIONAL COMPOUND NITTO DENKO CORPORATION (JP) 2011-04-28 US disclosed
US-20110046358-A1 METHOD FOR PRODUCTION OF POLYFUNCTIONAL COMPOUND NITTO DENKO CORPORATION (JP) 2011-02-24 US disclosed
US-7884167-B2 conducting a Michael addition of a compound (A) having a hydrogen atom of pKa less than or equal to 15 to a (meth)acrylate or a (meth)acrylamide (B), in which at least one of the compounds (A) and (B) has a photoisomerization group; optical recording material, optical waveguide material NITTO DENKO CORPORATION (JP) 2011-02-08 US disclosed
US-20100076216-A1 LIQUID CRYSTAL COMPOUND, OPTICAL ELEMENT, POLARIZING PLATE, IMAGE DISPLAY APPARATUS, AND OPTICAL RECORDING MATERIAL NITTO DENKO CORPORATION (JP) 2010-03-25 US disclosed
US-20090209741-A1 POLYFUNCTIONAL COMPOUND, OPTICAL RECORDING MATERIAL, OPTICAL RECORDING MEDIUM, OPTICAL RECORDING/REPRODUCING APPARATUS, OPTICAL WAVEGUIDE MATERIAL, AND PHOTO-ALIGNMENT FILM MATERIAL NITTO DENKO CORPORATION (JP) 2009-08-20 US disclosed
CN-101489993-A Method for producing polyfunctional compound NITTO DENKO CORP (JP) 2009-07-22 CN disclosed
US-20090182107-A1 METHOD FOR PRODUCTION OF POLYFUNCTIONAL COMPOUND NITTO DENKO CORPORATION (JP) 2009-07-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110046358-A1 METHOD FOR PRODUCTION OF POLYFUNCTIONAL COMPOUND ADCY10, ADCY5, ADCY1 FDPS 950/4885MEN1 646/4885AGTR1 4031/4885
US-20090209741-A1 POLYFUNCTIONAL COMPOUND, OPTICAL RECORDING MATERIAL, OPTICAL RECORDING MEDIUM, OPTICAL RECORDING/REPRODUCING APPARATUS, OPTICAL WAVEGUIDE MATERIAL, AND PHOTO-ALIGNMENT FILM MATERIAL CRY1, HAX1, F12 FDPS 4234/4885MEN1 720/4885AGTR1 2391/4885
US-20110098454-A1 METHOD FOR PRODUCTION OF POLYFUNCTIONAL COMPOUND ADCY10, ADCY5, ADCY1 FDPS 1057/4885MEN1 608/4885AGTR1 4036/4885
US-20100076216-A1 LIQUID CRYSTAL COMPOUND, OPTICAL ELEMENT, POLARIZING PLATE, IMAGE DISPLAY APPARATUS, AND OPTICAL RECORDING MATERIAL RCC1, NCAPD2, OCIAD1 FDPS 2303/4885MEN1 892/4885AGTR1 3303/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.