SCHEMBL13628854

SCHEMBL13628854

COOSc1ccc2c(c1)cc(Cc1nccs1)n2Cc1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.36
TP53 P04637 2/20 0.36
ALDH1A1 P00352 2/20 0.35
TSHR P16473 2/20 0.35
HSD17B10 Q99714 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
RECQL P46063 1/20 0.35
ALOX5AP P20292 2/20 0.34
THRB P10828 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
PARG Q86W56 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628821 0.83 MAPT (0.37) MAPTTP53ALDH1A1TSHRHSD17B10
SCHEMBL13628846 0.80 POLB (0.41) TP53ALDH1A1NPSR1HPGDLMNA
SCHEMBL2926901 0.79 PTGS2 (0.47) MAPTTP53ALDH1A1TSHRHSD17B10
SCHEMBL13628858 0.75 CCR2 (0.38) MAPTTP53TSHRNPSR1CYP1A2
SCHEMBL13628859 0.74 PTGS2 (0.45) TP53TBXA2RPOLB
SCHEMBL13628860 0.73 PTGS2 (0.46) MAPTTP53LMNATBXA2R
SCHEMBL13628851 0.71 PTGS2 (0.36) TP53ALDH1A1TSHRMEN1KMT2A
SCHEMBL13628847 0.71 CYP11B2 (0.43) MAPTNPSR1
SCHEMBL13628853 0.70 PTGS2 (0.37) MAPTALDH1A1TSHRKMT2ANPSR1
SCHEMBL13628824 0.69 RAB9A (0.36) MAPTALDH1A1TSHRMAPK1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed