SCHEMBL13680837

SCHEMBL13680837

CN(C)C(=O)c1ccc(-c2cccc(CCC=O)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.40
CYP3A4 P08684 5/20 0.40
CYP2D6 P10635 4/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
TP53 P04637 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HIF1A Q16665 1/20 0.40
CYP1A2 P05177 8/20 0.39
CLK4 Q9HAZ1 6/20 0.39
HSD17B10 Q99714 4/20 0.39
ERN1 O75460 4/20 0.39
ATR Q13535 3/20 0.39
CYP2C19 P33261 2/20 0.39
TSHR P16473 1/20 0.39
CYP2C9 P11712 2/20 0.39
USP2 O75604 2/20 0.38
MAPK1 P28482 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680825 0.87 MAPT (0.41) ALDH1A1HPGDKMT2AHSD17B10ATR
SCHEMBL13680830 0.84 RARA (0.44) ALDH1A1KDM4ETP53
SCHEMBL13680835 0.83 MAP4K4 (0.42) ERN1MAPK1
SCHEMBL15349861 0.82 ALDH1A1 (0.44) ALDH1A1CYP3A4CYP2D6KDM4EHPGD
SCHEMBL13680836 0.82 NPC1 (0.44) ATRHDAC4
SCHEMBL13680828 0.82 ALDH1A1 (0.42) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL13680842 0.81 RAB9A (0.45) ALDH1A1KDM4EHPGDKMT2ATSHR
SCHEMBL13680841 0.81 TSHR (0.40) KDM4EMEN1KMT2ATSHR
SCHEMBL13680831 0.81 PDE10A (0.37)
SCHEMBL13680834 0.79 PDE10A (0.39) ALDH1A1KDM4EHPGDTDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed