SCHEMBL154107

SCHEMBL154107

Cc1scccc(Cl)c(C)c(C)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.40
TSHR P16473 3/20 0.40
LMNA P02545 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
ALOX12 P18054 3/20 0.38
HPGD P15428 2/20 0.38
MAPT P10636 4/20 0.35
THRB P10828 1/20 0.35
POLB P06746 2/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
GAA P10253 4/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TP53 P04637 1/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL3327760 0.98 ALDH1A1 (0.39) ALDH1A1TSHRLMNASMN1; SMN2ALOX12
SCHEMBL4373436 0.91 ALDH1A1 (0.40) ALDH1A1TSHRLMNASMN1; SMN2ALOX12
SCHEMBL4369368 0.83 ALDH1A1 (0.40) ALDH1A1TSHRLMNASMN1; SMN2ALOX12
SCHEMBL5196982 0.74 TRPA1 (0.43) ALDH1A1TSHRLMNASMN1; SMN2HPGD
SCHEMBL150091 0.73 TSHR (0.41) ALDH1A1TSHRLMNASMN1; SMN2ALOX12
SCHEMBL10848388 0.69 ALDH1A1 (0.50) ALDH1A1TSHRLMNASMN1; SMN2ALOX12
SCHEMBL752673 0.68 TSHR (0.41) ALDH1A1TSHRSMN1; SMN2ALOX12HPGD
SCHEMBL112040 0.67
Hydrochloric Acid SCHEMBL31150435 0.67 TSHR (0.39) ALDH1A1TSHRSMN1; SMN2ALOX12HPGD
Hydrochloric Acid SCHEMBL154108 0.67 TSHR (0.39) ALDH1A1TSHRSMN1; SMN2ALOX12HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 229 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078142-A1 FULLY-CONTINUOUS SYNTHESIS METHOD OF CYPROTERONE ACETATE UNIV FUDAN (CN) 2026-03-19 US claimed
CN-102596967-B Prepare the photochemical method of Artemisinin SAI NUOFEI (FR) 2015-08-26 CN claimed
EP-2046767-B1 PROCESS FOR PREPARING DIAMINOPHENOTHIAZINIUM COMPOUNDS PROVENCE TECHNOLOGIES (FR) 2015-04-22 EP claimed
US-8765942-B2 Process for preparing diaminophenothiazinium compounds PROVENCE TECHNOLOGIES (FR) 2014-07-01 US claimed
US-20130299338-A1 PHOTOCHEMICAL PROCESS FOR PRODUCING ARTEMISININ SANOFI SA (FR) 2013-11-14 US claimed
US-8507697-B2 Photochemical process for producing artemisinin SANOFI (FR) 2013-08-13 US claimed
EP-2473512-A1 PHOTOCHEMICAL PROCESS FOR PRODUCING ARTEMISININ SANOFI (FR) 2012-07-11 EP claimed
US-20110250296-A1 REVERSE VITAMIN K EFFECT VIA PHOTODYNAMIC OXIDATION TARGETED AT VASCULAR ENDOTHELIUM, FIBRIN AND BLOOD PLATELETS WINSLOW DAVID E 2011-10-13 US claimed
US-7968127-B2 Reverse vitamin K effect via photodynamic oxidation targeted at vascular endothelium, fibrin and blood platelets WINSLOW DAVID E 2011-06-28 US claimed
US-20100021566-A1 REVERSE VITAMIN K EFFECT VIA PHOTODYNAMIC OXIDATION TARGETED AT VASCULAR ENDOTHELIUM, FIBRIN AND BLOOD PLATELETS WINSLOW DAVID E 2010-01-28 US claimed
US-20090291943-A1 PROCESS FOR PREPARING DIAMINOPHENOTHIAZINIUM COMPOUNDS PROVEPHARM LIFE SOLUTIONS (FR) 2009-11-26 US claimed
EP-4017496-B1 FORMULATIONS FOR USE IN THE PREVENTION AND/OR TREATMENT OF PERIPHERAL NEUROPATHY AND ITS ASSOCIATED DISEASES LOH YIN SZE (SG) 2026-01-07 EP disclosed
US-20250325557-A1 3, 7-DIAMINO-10H-PHENOTHIAZINE SALTS AND THEIR USE WISTA LABORATORIES LTD. (SG) 2025-10-23 US disclosed
US-20250222006-A1 METHODS OF SYNTHESIS AND/OR PURIFICATION OF DIAMINOPHENOTHIAZINIUM COMPOUNDS WISTA LABORATORIES LTD. (SG) 2025-07-10 US disclosed
EP-3795565-B1 IMPROVED PROCESS FOR THE PURIFICATION OF METHYLENE BLUE RK PHARMA INC (US) 2025-07-09 EP disclosed
US-6022549-A NONAQUEOUS, COMPRISING A PHENOL ANTIMICROBIAL AGENT, A FILM FORMING RESIN, AND ORGANIC SOLVENT; THE PHENOL IS STORAGE STABLE AND CAPABLE OF LEACHING FOLLOWING SOLIDIFICATION OF THE NAIL COATING WITHOUT LOSING MICROBIOCIDAL ACTIVITY WOODWARD LABORATORIES, INC. (US) 2000-02-08 US disclosed
US-6013677-A APPLYING TO THE NAIL A NON-AQUEOUS ANTIMICROBIAL NAIL COATING CONTAINING A FILM FORMING POLYMER, AN ORGANIC SOLVENT, A ANTIMICROBIAL AGENT COMPRISING SOLUBILZED BENZALKONIUM CHLORIDE AND CAPABLE OF LEACHING FROM NAIL COATING WOODWARD LABORATORIES, INC. (US) 2000-01-11 US disclosed
US-5968986-A NONAQUEOUS NAIL COATING WITH MICROBIOCDES AND POLYMERS WOODWARD LABORATORIES, INC. (US) 1999-10-19 US disclosed
US-5961469-A Spectrophotometric assay for cyanide ROIZEN MICHAEL F (US) 1999-10-05 US disclosed
WO-1999036033-A1 ANTIMICROBIAL NAIL COATING COMPOSITION WOODWARD LABORATORIES, INC. (US) 1999-07-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250325557-A1 3, 7-DIAMINO-10H-PHENOTHIAZINE SALTS AND THEIR USE PSEN1, PSEN2, APP ALDH1A1 2648/4885TSHR 1453/4885LMNA 222/4885
US-20250222006-A1 METHODS OF SYNTHESIS AND/OR PURIFICATION OF DIAMINOPHENOTHIAZINIUM COMPOUNDS MB, TPMT, HBB ALDH1A1 1477/4885TSHR 1603/4885LMNA 2166/4885
US-20100021566-A1 REVERSE VITAMIN K EFFECT VIA PHOTODYNAMIC OXIDATION TARGETED AT VASCULAR ENDOTHELIUM, FIBRIN AND BLOOD PLATELETS PROC, PFKP, TTPA ALDH1A1 2051/4885TSHR 3001/4885LMNA 2440/4885
US-20110250296-A1 REVERSE VITAMIN K EFFECT VIA PHOTODYNAMIC OXIDATION TARGETED AT VASCULAR ENDOTHELIUM, FIBRIN AND BLOOD PLATELETS PROC, PFKP, TTPA ALDH1A1 2051/4885TSHR 3001/4885LMNA 2440/4885
US-20130299338-A1 PHOTOCHEMICAL PROCESS FOR PRODUCING ARTEMISININ DHPS, FDPS, GGPS1 ALDH1A1 559/4885TSHR 4498/4885LMNA 2799/4885
US-20090291943-A1 PROCESS FOR PREPARING DIAMINOPHENOTHIAZINIUM COMPOUNDS DCPS, QDPR, DNPEP ALDH1A1 1379/4885TSHR 3603/4885LMNA 2709/4885
US-20260078142-A1 FULLY-CONTINUOUS SYNTHESIS METHOD OF CYPROTERONE ACETATE CYP17A1, CYP21A2, HSD17B2 ALDH1A1 241/4885TSHR 456/4885LMNA 2995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.